SCHEMBL4690738

SCHEMBL4690738

Cc1ccc(C(=O)N2CC3CN(C(CC(N)=O)c4ccc(C)c(Cl)c4)CC3C2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 10/20 0.46
HCRTR2 O43614 10/20 0.46
HPGD P15428 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TNF P01375 1/20 0.36
P2RX7 Q99572 2/20 0.34
UTS2R Q9UKP6 1/20 0.34
MGLL Q99685 1/20 0.33
PDE2A O00408 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4695935 0.93 HCRTR2 (0.47) HCRTR1HCRTR2HPGDALDH1A1TNF
SCHEMBL4694375 0.90 HCRTR1 (0.40) HCRTR1HCRTR2HPGDALDH1A1TNF
SCHEMBL4692886 0.89 ALDH1A1 (0.42) HCRTR1HCRTR2HPGDALDH1A1TNF
SCHEMBL4690927 0.89 HCRTR1 (0.49) HCRTR1HCRTR2ALDH1A1MGLLLMNA
SCHEMBL4690680 0.89 HCRTR1 (0.42) HCRTR1HCRTR2HPGDALDH1A1TNF
SCHEMBL4694334 0.88 HCRTR1 (0.43) HCRTR1HCRTR2TNF
SCHEMBL4692692 0.86 HCRTR1 (0.45) HCRTR1HCRTR2ALDH1A1TNFPDE2A
SCHEMBL4690403 0.86 HCRTR1 (0.39) HCRTR1HCRTR2HPGDALDH1A1TNF
SCHEMBL4692944 0.86 HCRTR1 (0.41) HCRTR1HCRTR2ALDH1A1P2RX7KDM4E
SCHEMBL4694969 0.86 HCRTR1 (0.38) HCRTR1HCRTR2HPGDTNFP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed