SCHEMBL4695050

SCHEMBL4695050

Cc1noc(C)c1S(=O)(=O)N1CC2CN(CC[C@H](N)c3ccccc3)CC2C1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.53
LMNA P02545 2/20 0.53
ALDH1A1 P00352 2/20 0.52
HTT P42858 1/20 0.51
CCR5 P51681 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
GFER P55789 1/20 0.42
PKM P14618 1/20 0.42
CHRM1 P11229 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
USP2 O75604 1/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4691491 0.81 FPR2 (0.50) ALDH1A1
SCHEMBL4691441 0.80 CCR5 (0.67) TSHRLMNAALDH1A1CCR5MEN1
SCHEMBL4689791 0.80 EPHX2 (0.49) ALDH1A1CCR5MEN1KMT2A
SCHEMBL4691597 0.80 FPR2 (0.47) ALDH1A1CCR5
SCHEMBL4692842 0.77 GBA1 (0.43) ALDH1A1CCR5KMT2AUSP2POLB
SCHEMBL4696460 0.74 CCR5 (0.51) TSHRLMNAALDH1A1CCR5MEN1
SCHEMBL4691646 0.74 LMNA (0.59) TSHRLMNAALDH1A1HTTCCR5
SCHEMBL4694247 0.72 DRD2 (0.36) ALDH1A1CCR5MAPK1
SCHEMBL3282872 0.72 DRD2 (0.36) ALDH1A1CCR5MAPK1
SCHEMBL4691804 0.72 CCR5 (0.47) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP claimed
EP-1761542-B1 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS HOFFMANN LA ROCHE (CH) 2008-01-02 EP disclosed