SCHEMBL4699124

SCHEMBL4699124

O=C1OCCC1CSCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.54
KCNH3 Q9ULD8 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAPK1 P28482 1/20 0.38
MC4R P32245 1/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3685687 0.78 MAOB (0.49) CRBNKCNH3
SCHEMBL7906013 0.78 MAOB (0.49) CRBNKCNH3
SCHEMBL7899581 0.78 MAOB (0.49) CRBNKCNH3
SCHEMBL11870917 0.76 FASN (0.45) KCNH3
SCHEMBL7767198 0.74 CRBN (0.49) CRBNL3MBTL1ALDH1A1LMNAHTT
SCHEMBL30226689 0.72 LMNA (0.48) KCNH3LMNAKMT2A
SCHEMBL3385520 0.72 KCNH3 (0.42) KCNH3L3MBTL1KMT2AMAPT
SCHEMBL7764865 0.70 CRBN (0.45) CRBNL3MBTL1ALDH1A1LMNAHTT
SCHEMBL25131268 0.70 KCNH3 (0.43) KCNH3ALDH1A1LMNASMN1; SMN2
SCHEMBL566956 0.70 CRBN (0.42) CRBNL3MBTL1ALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444202-B1 NOVEL METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2008-10-15 EP disclosed
US-7132434-B2 Metalloproteinase inhibitors ASTRAZENECA AB (SE) 2006-11-07 US disclosed
US-20050026990-A1 Novel metalloproteinase ihibitors ASTRAZENECA AB (SE) 2005-02-03 US disclosed
EP-1444202-A1 NOVEL METALLOPROTEINASE INHIBITORS AstraZeneca AB (SE) 2004-08-11 EP disclosed
WO-2003040098-A1 NOVEL METALLOPROTEINASE INHIBITORS ASTRAZENECA AB (SE) 2003-05-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050026990-A1 Novel metalloproteinase ihibitors MMP12, MMP1, MMP16 CRBN 1675/4885KCNH3 4078/4885L3MBTL1 3869/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.