SCHEMBL4699567

SCHEMBL4699567

CC(C)C[C@@H](C(N)=O)N(CC#N)c1cscc1-c1ccc(N2CCN(C)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.44
CTSB P07858 9/20 0.44
CTSS P25774 9/20 0.44
CTSL P07711 8/20 0.44
HDAC3 O15379 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
RPS6KA3 P51812 1/20 0.37
ABL1 P00519 1/20 0.35
LCK P06239 1/20 0.35
RET P07949 1/20 0.35
HCK P08631 1/20 0.35
KIT P10721 1/20 0.35
SRC P12931 1/20 0.35
PDGFRA P16234 1/20 0.35
KDR P35968 1/20 0.35
TEK Q02763 1/20 0.35
PRKD1 Q15139 1/20 0.35
CHEK1 O14757 1/20 0.34
GRM2 Q14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756631 0.88 RET (0.40) RET
SCHEMBL4703612 0.83 CTSS (0.34) CTSKCTSBCTSSCTSL
SCHEMBL4701830 0.82 CTSK (0.37) CTSKCTSBCTSSCTSL
SCHEMBL4703746 0.82 OPRM1 (0.37) CTSKCTSBCTSSCTSLCHEK1
SCHEMBL4704896 0.80 CTSK (0.34) CTSKCTSBCTSSCTSL
SCHEMBL4704688 0.80 CTSL (0.33) CTSKCTSBCTSSCTSL
SCHEMBL4699887 0.79 CTSS (0.34) CTSKCTSBCTSSCTSL
SCHEMBL4703317 0.79 HRH3 (0.35) CTSKCTSBCTSSCTSL
SCHEMBL4704824 0.79 CTSK (0.36) CTSKCTSBCTSSCTSL
SCHEMBL4703639 0.79 CTSK (0.36) CTSKCTSBCTSSCTSLPRKD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed