SCHEMBL4703746

SCHEMBL4703746

CC(C)C[C@@H](C(N)=O)N(CC#N)c1cscc1-c1ccc(CN2CCCC2)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.37
OPRK1 P41145 1/20 0.37
HRH3 Q9Y5N1 8/20 0.36
CHKA P35790 2/20 0.36
ACACB O00763 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
MCHR1 Q99705 2/20 0.35
ALDH1A1 P00352 1/20 0.34
CHEK1 O14757 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
TBK1 Q9UHD2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4704801 0.92 HRH3 (0.37) HRH3CTSLCTSBCTSSCTSK
SCHEMBL4703463 0.86 HRH3 (0.37) OPRM1OPRK1HRH3CTSLCTSB
SCHEMBL4701956 0.86 SPHK1 (0.39) HRH3CTSLCTSBCTSSCTSK
SCHEMBL4703639 0.84 CTSK (0.36) CTSLCTSBCTSSCTSK
SCHEMBL4704688 0.84 CTSL (0.33) HRH3CTSLCTSBCTSSCTSK
SCHEMBL4704896 0.84 CTSK (0.34) CTSLCTSBCTSSCTSK
SCHEMBL4703317 0.83 HRH3 (0.35) HRH3CTSLCTSBCTSSCTSK
SCHEMBL4703612 0.83 CTSS (0.34) CTSLCTSBCTSSCTSK
SCHEMBL4703525 0.82 AGTR2 (0.40)
SCHEMBL4701830 0.82 CTSK (0.37) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed