SCHEMBL4700607

SCHEMBL4700607

CC(C)C[C@H](N)C(=O)N(CC#N)c1cscc1-c1ccc(CNCc2ccccc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 2/20 0.37
CTSK P43235 6/20 0.36
CTSB P07858 4/20 0.36
CTSS P25774 3/20 0.36
CTSL P07711 2/20 0.36
ANPEP P15144 2/20 0.34
HDAC1 Q13547 1/20 0.33
RNPEP Q9H4A4 1/20 0.33
DNPEP Q9ULA0 1/20 0.33
CIT O14578 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CTSH P09668 1/20 0.32
CYP2D6 P10635 1/20 0.32
CTSC P53634 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703749 0.87 CTSK (0.32) CTSKCTSBCTSSCTSL
SCHEMBL4701046 0.82 AKR1C3 (0.34) GPR88CTSKCTSBCTSSCTSL
SCHEMBL4701072 0.75 PDCD1 (0.35) CTSKCTSBCTSSCTSLSMN1; SMN2
SCHEMBL4704896 0.74 CTSK (0.34) CTSKCTSBCTSSCTSL
SCHEMBL4701624 0.74 CTSL (0.42) CTSBCTSSCTSL
SCHEMBL4699471 0.73 KCNH2 (0.36) CTSKCTSBCTSSCTSL
SCHEMBL4703639 0.73 CTSK (0.36) CTSKCTSBCTSSCTSL
SCHEMBL4701830 0.72 CTSK (0.37) GPR88CTSKCTSBCTSSCTSL
SCHEMBL4699453 0.71 CTSS (0.64) CTSKCTSBCTSSCTSL
SCHEMBL4703463 0.69 HRH3 (0.37) CTSKCTSBCTSSCTSLHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed