SCHEMBL4702622

SCHEMBL4702622

CC(C)C[C@@H](C(N)=O)N(CC#N)c1cscc1-c1cccc(CO)c1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.33
CTSK P43235 6/20 0.32
CTSS P25774 5/20 0.32
CTSL P07711 5/20 0.32
PI4K2A Q9BTU6 1/20 0.32
CTSB P07858 2/20 0.32
PIP4K2A P48426 1/20 0.31
CTSA P10619 1/20 0.31
LRRK2 Q5S007 1/20 0.31
HPGDS O60760 1/20 0.31
ADAMTS4 O75173 1/20 0.31
PRKCI P41743 1/20 0.30
CTSD P07339 1/20 0.30
MMP1 P03956 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703269 0.91 ATP4A (0.36) CTSKCTSSCTSLMMP1
SCHEMBL4701830 0.89 CTSK (0.37) CTSKCTSSCTSLCTSBMMP1
SCHEMBL6801548 0.88 CTSS (0.35) CTSKCTSSCTSLCTSBHPGDS
SCHEMBL4701371 0.83 CTSL (0.33) CTSKCTSSCTSLCTSB
SCHEMBL4703612 0.83 CTSS (0.34) CTSKCTSSCTSLCTSB
SCHEMBL4704688 0.82 CTSL (0.33) CTSKCTSSCTSLCTSB
SCHEMBL4704896 0.82 CTSK (0.34) CTSKCTSSCTSLCTSB
SCHEMBL4703317 0.82 HRH3 (0.35) CTSKCTSSCTSLCTSB
SCHEMBL4703639 0.81 CTSK (0.36) CTSKCTSSCTSLCTSB
SCHEMBL4699887 0.80 CTSS (0.34) CTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1372655-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-10-01 EP disclosed