SCHEMBL470845

SCHEMBL470845

CCc1cc(C)cnc1Oc1ccc(N)c(NC)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 2/20 0.36
ATP4B P51164 2/20 0.36
DRD1 P21728 3/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
PTGER4 P35408 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SLC13A5 Q86YT5 1/20 0.31
CDK8 P49336 1/20 0.31
AOC1 P19801 1/20 0.31
AOC3 Q16853 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470990 0.85 NOS3 (0.38) DRD1PTGER4NOS3NOS1NOS2
SCHEMBL471096 0.83 BACE1 (0.40) DRD1PTGER4BACE1BACE2
SCHEMBL10005546 0.81 DRD1 (0.33) DRD1NOS3NOS1MAPTALDH1A1
SCHEMBL470986 0.75 DRD1 (0.45) DRD1SLC6A4PTGER4ALDH1A1BACE1
SCHEMBL470989 0.75 DRD1 (0.46) DRD1SLC6A2SLC6A4PTGER4CDK8
SCHEMBL470941 0.74 SMN1; SMN2 (0.60) DRD1L3MBTL1
SCHEMBL13211386 0.73 NR4A1 (0.54) KMT2AMEN1HTTMAPTALDH1A1
SCHEMBL471097 0.73 AGXT (0.36) ATP4AATP4BDRD1KMT2AMEN1
SCHEMBL10005544 0.72 LTA4H (0.45) DRD1BACE1BACE2
SCHEMBL470868 0.71 NR4A1 (0.34) DRD1KMT2AMEN1NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033091-A1 PROCESS FOR PREPARING BENZOIC ACID ESTERS 第一三共株式会社 (JP) 2012-03-15 WO disclosed
WO-2010101164-A1 PYRIDINE DERIVATIVE 第一三共株式会社 (JP) 2010-09-10 WO disclosed