SCHEMBL471096

SCHEMBL471096

CNc1cc(Oc2ncc(C)cc2F)ccc1N

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.40
BACE2 Q9Y5Z0 8/20 0.40
PPARG P37231 1/20 0.37
PTGER4 P35408 1/20 0.36
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4D Q08499 1/20 0.33
TRPA1 O75762 1/20 0.33
EGLN1 Q9GZT9 1/20 0.32
DRD1 P21728 1/20 0.32
LTA4H P09960 2/20 0.32
KCNH2 Q12809 1/20 0.32
LYN P07948 1/20 0.31
BTK Q06187 1/20 0.31
NR4A1 P22736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470990 0.86 NOS3 (0.38) PPARGPTGER4DRD1NR4A1
SCHEMBL10005544 0.86 LTA4H (0.45) BACE1BACE2PPARGTRPA1DRD1
SCHEMBL470845 0.83 ATP4A (0.36) BACE1BACE2PTGER4DRD1
SCHEMBL470986 0.82 DRD1 (0.45) BACE1BACE2PPARGPTGER4PDE4A
SCHEMBL470989 0.76 DRD1 (0.46) PPARGPTGER4DRD1
SCHEMBL471003 0.76 TRPA1 (0.34) BACE1BACE2TRPA1NR4A1
SCHEMBL470941 0.75 SMN1; SMN2 (0.60) PPARGDRD1
SCHEMBL13211386 0.74 NR4A1 (0.54) NR4A1
SCHEMBL471097 0.74 AGXT (0.36) DRD1KCNH2
SCHEMBL10005546 0.74 DRD1 (0.33) EGLN1DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033091-A1 PROCESS FOR PREPARING BENZOIC ACID ESTERS 第一三共株式会社 (JP) 2012-03-15 WO disclosed
WO-2010101164-A1 PYRIDINE DERIVATIVE 第一三共株式会社 (JP) 2010-09-10 WO disclosed