SCHEMBL470990

SCHEMBL470990

CNc1cc(Oc2ncc(C)cc2C)ccc1N

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
PPARG P37231 1/20 0.35
DRD1 P21728 4/20 0.35
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
NR4A1 P22736 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP2A6 P11509 1/20 0.32
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
PTGER4 P35408 1/20 0.31
SCN9A Q15858 1/20 0.30
LMNA P02545 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
APEX1 P27695 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CDK8 P49336 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL471096 0.86 BACE1 (0.40) PPARGDRD1NR4A1PTGER4
SCHEMBL470989 0.86 DRD1 (0.46) PPARGDRD1KDM4EPOLBPTGER4
SCHEMBL470986 0.86 DRD1 (0.45) PPARGDRD1KDM4EPOLBNR4A1
SCHEMBL470845 0.85 ATP4A (0.36) NOS3NOS1NOS2DRD1ALDH1A1
SCHEMBL10005546 0.84 DRD1 (0.33) NOS3NOS1DRD1KDM4EPOLB
SCHEMBL470868 0.80 NR4A1 (0.34) NOS3NOS1NOS2DRD1NR4A1
SCHEMBL471097 0.79 AGXT (0.36) DRD1KDM4EPOLBALDH1A1LMNA
SCHEMBL470941 0.77 SMN1; SMN2 (0.60) PPARGDRD1LMNACYP2C9TSHR
SCHEMBL13211386 0.77 NR4A1 (0.54) KDM4EPOLBNR4A1ALDH1A1TSHR
SCHEMBL10005544 0.75 LTA4H (0.45) PPARGDRD1LMNACYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033091-A1 PROCESS FOR PREPARING BENZOIC ACID ESTERS 第一三共株式会社 (JP) 2012-03-15 WO disclosed
WO-2010101164-A1 PYRIDINE DERIVATIVE 第一三共株式会社 (JP) 2010-09-10 WO disclosed