SCHEMBL470989

SCHEMBL470989

CNc1cc(Oc2ncc(Cl)cc2C)ccc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 3/20 0.46
CYP2C9 P11712 2/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
APEX1 P27695 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MAPK1 P28482 1/20 0.40
EGFR P00533 1/20 0.38
PPARG P37231 1/20 0.37
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
SCN9A Q15858 2/20 0.36
LIPE Q05469 3/20 0.34
BCHE P06276 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CDK8 P49336 1/20 0.33
SCN5A Q14524 1/20 0.33
CHUK O15111 1/20 0.33
CCR2 P41597 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470941 0.88 SMN1; SMN2 (0.60) DRD1CYP2C9LMNATSHRAPEX1
SCHEMBL470990 0.86 NOS3 (0.38) DRD1CYP2C9LMNATSHRAPEX1
SCHEMBL10005544 0.86 LTA4H (0.45) DRD1CYP2C9LMNATSHRAPEX1
SCHEMBL470986 0.84 DRD1 (0.45) DRD1PPARGKDM4EPOLBSLC6A4
SCHEMBL10005546 0.82 DRD1 (0.33) DRD1SMN1; SMN2KDM4EPOLB
SCHEMBL470868 0.78 NR4A1 (0.34) DRD1SMN1; SMN2SCN9A
SCHEMBL471097 0.77 AGXT (0.36) DRD1CYP2C9LMNATSHRAPEX1
SCHEMBL471096 0.76 BACE1 (0.40) DRD1PPARGPTGER4
SCHEMBL470845 0.75 ATP4A (0.36) DRD1SLC6A2SLC6A4CDK8PTGER4
SCHEMBL13211386 0.74 NR4A1 (0.54) TSHRSMN1; SMN2MAPK1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033091-A1 PROCESS FOR PREPARING BENZOIC ACID ESTERS 第一三共株式会社 (JP) 2012-03-15 WO disclosed
WO-2010101164-A1 PYRIDINE DERIVATIVE 第一三共株式会社 (JP) 2010-09-10 WO disclosed