SCHEMBL470986

SCHEMBL470986

CNc1cc(Oc2ncc(F)cc2C)ccc1N

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 4/20 0.45
PPARG P37231 1/20 0.37
BACE1 P56817 5/20 0.35
BACE2 Q9Y5Z0 5/20 0.35
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4D Q08499 1/20 0.33
SLC6A4 P31645 1/20 0.33
PTGER4 P35408 3/20 0.32
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
GCK P35557 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NR4A1 P22736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL470990 0.86 NOS3 (0.38) DRD1PPARGPTGER4KDM4EPOLB
SCHEMBL470989 0.84 DRD1 (0.46) DRD1PPARGSLC6A4PTGER4KDM4E
SCHEMBL10005546 0.82 DRD1 (0.33) DRD1KDM4EPOLBALDH1A1
SCHEMBL471096 0.82 BACE1 (0.40) DRD1PPARGBACE1BACE2PDE4A
SCHEMBL10005544 0.78 LTA4H (0.45) DRD1PPARGBACE1BACE2
SCHEMBL470868 0.78 NR4A1 (0.34) DRD1ALDH1A1NR4A1
SCHEMBL471097 0.77 AGXT (0.36) DRD1KDM4EPOLBALDH1A1
SCHEMBL470845 0.75 ATP4A (0.36) DRD1BACE1BACE2SLC6A4PTGER4
SCHEMBL30166991 0.75 HDAC1 (0.47) PDE4APDE4BPDE4DKDM4EGCK
SCHEMBL470941 0.75 SMN1; SMN2 (0.60) DRD1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033091-A1 PROCESS FOR PREPARING BENZOIC ACID ESTERS 第一三共株式会社 (JP) 2012-03-15 WO disclosed
WO-2010101164-A1 PYRIDINE DERIVATIVE 第一三共株式会社 (JP) 2010-09-10 WO disclosed