SCHEMBL4709657

SCHEMBL4709657

CC(c1ccccc1Cl)N1CCN=C1c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1N1CCOCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
TACR1 P25103 3/20 0.34
HPGD P15428 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
CNR2 P34972 1/20 0.32
CETP P11597 2/20 0.32
SOS1 Q07889 2/20 0.32
TSHR P16473 2/20 0.31
GAA P10253 2/20 0.31
KDM4E B2RXH2 1/20 0.31
PIK3CD O00329 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
HTT P42858 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MAPT P10636 1/20 0.31
NR4A1 P22736 1/20 0.31
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
DPP4 P27487 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705055 0.84 ALDH1A1 (0.34) ALDH1A1TACR1HPGDSMN1; SMN2CNR2
SCHEMBL4705320 0.83 SOS1 (0.34) ALDH1A1TACR1HPGDSMN1; SMN2CNR2
SCHEMBL4706657 0.83 ALDH1A1 (0.42) ALDH1A1TACR1HPGDSMN1; SMN2CNR2
SCHEMBL4705321 0.82 TACR1 (0.35) ALDH1A1TACR1HPGDSMN1; SMN2TSHR
SCHEMBL4708876 0.76 GHSR (0.38) ALDH1A1TACR1HPGDSMN1; SMN2TSHR
Hydrochloric Acid SCHEMBL4708409 0.73 LMNA (0.36) TACR1HPGDSMN1; SMN2CETPTSHR
SCHEMBL4705280 0.73 PTGER4 (0.40) TACR1
SCHEMBL4790291 0.73 PTGER4 (0.40) TACR1
SCHEMBL4707556 0.73 RORB (0.39) ALDH1A1SMN1; SMN2TSHRKDM4EPIK3CA
SCHEMBL4706503 0.70 P2RX7 (0.37) ALDH1A1HPGDSMN1; SMN2TSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501809-B1 TRIAZOLE DERIVATIVES AS TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-01-16 EP disclosed