SCHEMBL4717868

SCHEMBL4717868

CC(C)Oc1ccc(C(=O)NNC(=O)N(C)Cc2ccc3nc(-c4ccccc4)[nH]c3c2)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 5/20 0.46
HDAC1 Q13547 5/20 0.46
HDAC8 Q9BY41 5/20 0.46
HDAC6 Q9UBN7 5/20 0.46
HDAC2 Q92769 3/20 0.46
CENPE Q02224 1/20 0.46
CHEK2 O96017 3/20 0.44
IKBKB O14920 1/20 0.43
SCD O00767 3/20 0.42
ITGB1 P05556 1/20 0.41
ITGA4 P13612 1/20 0.41
ITGB7 P26010 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2617481 0.85 CHEK2 (0.47) HDAC3HDAC1HDAC8HDAC6HDAC2
SCHEMBL4721149 0.84 CENPE (0.55) CENPE
SCHEMBL4717871 0.81 CENPE (0.43) HDAC3HDAC1HDAC8HDAC6HDAC2
SCHEMBL2107051 0.79 CENPE (0.47) HDAC3HDAC1HDAC8HDAC6HDAC2
SCHEMBL4720085 0.78 CENPE (0.54) HDAC1HDAC8HDAC6CENPE
SCHEMBL4718071 0.78 CENPE (0.49) HDAC3HDAC1HDAC2CENPE
SCHEMBL4720907 0.77 TRPM8 (0.50) HDAC1HDAC8HDAC6HDAC2CENPE
SCHEMBL4720148 0.77 PTGES (0.52) HDAC1HDAC8HDAC6CENPE
SCHEMBL4720774 0.77 CENPE (0.47) CENPE
SCHEMBL2617484 0.77 HPSE (0.46) HDAC3HDAC1HDAC8HDAC6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed