SCHEMBL4720148

SCHEMBL4720148

CC(C)Oc1ccc(C(=O)NNC(=O)N(C)Cc2cccc(OCc3ccccc3)c2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.52
CENPE Q02224 1/20 0.47
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
KMT2A Q03164 4/20 0.43
SMPD1 P17405 1/20 0.43
CTSK P43235 1/20 0.43
GPR132 Q9UNW8 1/20 0.43
MEN1 O00255 3/20 0.43
NR1H4 Q96RI1 1/20 0.42
LTB4R Q15722 1/20 0.42
LTB4R2 Q9NPC1 1/20 0.42
MRGPRX4 Q96LA9 3/20 0.42
CYP19A1 P11511 1/20 0.42
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4718071 0.92 CENPE (0.49) PTGESCENPEHDAC1KMT2ACTSK
SCHEMBL4720907 0.88 TRPM8 (0.50) CENPEHDAC1HDAC8HDAC6KMT2A
SCHEMBL2103625 0.84 PTGES (0.48) PTGESCENPEHDAC1HDAC8HDAC6
SCHEMBL4721149 0.84 CENPE (0.55) CENPEKMT2ASMPD1MEN1
SCHEMBL4720085 0.82 CENPE (0.54) PTGESCENPEHDAC1HDAC8HDAC6
SCHEMBL4720774 0.80 CENPE (0.47) CENPEKMT2ASMPD1MEN1POLB
SCHEMBL4721235 0.79 CENPE (0.44) PTGESCENPEHDAC1KMT2AMEN1
SCHEMBL4720150 0.79 PTGES (0.46) PTGESCENPEHDAC1HDAC8HDAC6
SCHEMBL2617475 0.78 HDAC3 (0.51) CENPEHDAC1KMT2AMEN1POLB
SCHEMBL4717868 0.77 HDAC3 (0.46) CENPEHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed