SCHEMBL4721149

SCHEMBL4721149

CC(C)Oc1ccc(C(=O)NNC(=O)N(C)Cc2ccc(-c3ccccc3)cc2)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 2/20 0.55
KIFC1 Q9BW19 1/20 0.50
CYP3A4 P08684 1/20 0.46
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 3/20 0.43
S1PR1 P21453 2/20 0.43
HPGD P15428 1/20 0.43
S1PR3 Q99500 1/20 0.43
SMPD1 P17405 1/20 0.41
ROCK2 O75116 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
LMNA P02545 1/20 0.40
MCHR1 Q99705 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4720085 0.90 CENPE (0.54) CENPEKMT2AMEN1HPGDROCK2
SCHEMBL4718071 0.89 CENPE (0.49) CENPEKMT2AMEN1CYP1A2CYP2C9
SCHEMBL4720774 0.88 CENPE (0.47) CENPEKIFC1KMT2AMEN1ALDH1A1
SCHEMBL4720907 0.85 TRPM8 (0.50) CENPECYP3A4KMT2AMEN1CYP1A2
SCHEMBL4720148 0.84 PTGES (0.52) CENPEKMT2AMEN1SMPD1
SCHEMBL4717868 0.84 HDAC3 (0.46) CENPE
SCHEMBL2103268 0.82 CENPE (0.56) CENPEKIFC1CYP3A4KMT2AMEN1
SCHEMBL2104964 0.81 CENPE (0.53) CENPEKIFC1CYP3A4KMT2AMEN1
SCHEMBL2101902 0.81 CENPE (0.51) CENPEKIFC1CYP3A4KMT2AMEN1
SCHEMBL5569249 0.79 CENPE (0.48) CENPEKIFC1KMT2AMEN1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1951719-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-08-06 EP disclosed
WO-2007056469-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed