SCHEMBL472949

SCHEMBL472949

CC1(C)C(C=O)C1C(=O)OCc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
LMNA P02545 2/20 0.58
ADRA2A P08913 1/20 0.58
CNR1 P21554 1/20 0.58
ATM Q13315 1/20 0.58
ALDH1A1 P00352 3/20 0.47
FABP7 O15540 1/20 0.44
FABP5 Q01469 1/20 0.44
HCAR2 Q8TDS4 1/20 0.43
ELANE P08246 3/20 0.43
MAPK1 P28482 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KMT2A Q03164 1/20 0.42
GAA P10253 1/20 0.42
PKM P14618 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6054965 0.90 TDP1 (0.64) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL3681483 0.87 TDP1 (0.57) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL3681480 0.87 TDP1 (0.57) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL1539179 0.86 TDP1 (0.80) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL1074161 0.86 TDP1 (0.63) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL1072275 0.86 TDP1 (0.54) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL1074157 0.86 TDP1 (0.63) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL22931582 0.86 TDP1 (0.76) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL523193 0.86 TDP1 (0.76) TDP1L3MBTL1LMNAADRA2ACNR1
SCHEMBL4433235 0.86 TDP1 (0.76) TDP1L3MBTL1LMNAADRA2ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2412702-B1 METHOD FOR PRODUCING CYCLOPROPANECARBOXYLIC ACID ESTER SUMITOMO CHEMICAL CO (JP) 2014-12-03 EP disclosed
EP-1970369-B1 METHOD FOR PRODUCING PURIFIED FORMYLCYCLOPROPANE COMPOUND AND INTERMEDIATE OF SUCH FORMYLCYCLOPROPANE COMPOUND SUMITOMO CHEMICAL CO (JP) 2013-09-25 EP disclosed
US-8263797-B2 Method for producing cyclopropane carboxylic acid compound and intermediate therefor SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-09-11 US disclosed
US-8168816-B2 Method for producing purified formylcyclopropane compound and intermediate of such formylcyclopropane compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-05-01 US disclosed
EP-1535895-B1 PROCESS FOR PRODUCTION OF FORMYLCYCLOPROPANECARBOXYLIC ESTERS SUMITOMO CHEMICAL CO (JP) 2012-04-25 EP disclosed
US-20120029227-A1 METHOD FOR PRODUCING CYCLOPROPANECARBOXYLIC ACID ESTER SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-02-02 US disclosed
EP-2412702-A1 METHOD FOR PRODUCING CYCLOPROPANECARBOXYLIC ACID ESTER Sumitomo Chemical Company, Limited (JP) 2012-02-01 EP disclosed
EP-1609776-B1 PROCESS FOR PRODUCTION OF CARBONYL COMPOUNDS SUMITOMO CHEMICAL CO (JP) 2011-03-02 EP disclosed
US-20100305353-A1 METHOD FOR PRODUCING PURIFIED FORMYLCYCLOPROPANE COMPOUND AND INTERMEDIATE OF SUCH FORMYLCYCLOPROPANE COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-12-02 US disclosed
US-20100280267-A1 METHOD FOR PRODUCING CYCLOPROPANE CARBOXYLIC ACID COMPOUND AND INTERMEDIATE THEREFOR SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2010-11-04 US disclosed
WO-2003066559-A1 PROCESS FOR PRODUCTION OF ALDEHYDES AND KETONES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-08-14 WO disclosed
WO-2003066566-A1 PROCESS FOR THE PRODUCTION OF TRANS-3,3-DIMETHYL-2-FORMLCYCLOPROPANE CARBOXYLIC ACID ESTERS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-08-14 WO disclosed
WO-2003059861-A1 PROCESS FOR PRODUCTION OF 3,3-DIMETHYL-2-FORMYLCYCLOPROPANECARBOXYLIC ACID DERIVATIVES SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2003-07-24 WO disclosed
US-6489505-B2 REACTING CHRYSANTHEMIC ACID ESTER WITH HYDROGEN PEROXIDE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-12-03 US disclosed
EP-1188735-A1 Process for producing carbonyl or hydroxy compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-03-20 EP disclosed
US-20020025906-A1 Process for producing carbonyl or hydroxy compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-02-28 US disclosed
US-20020010361-A1 Process for producing 3,3-dimethyl-2- formylcyclopropane-carboxylic acid ester SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2002-01-24 US disclosed
EP-1120393-A1 A process for producing 3,3-dimethyl-2-formylcyclopropane-carboxylic acid ester SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2001-08-01 EP disclosed
US-4864052-A 2,2-Dimethylcyclopropane-carboxylic acid derivatives SAGAMI CHEMICAL RESEARCH CENTER (JP) 1989-09-05 US disclosed
EP-0217342-A1 2,2-Dimethylcyclopropanecarboxylic acid derivatives SAGAMI CHEMICAL RESEARCH CENTER (JP) 1987-04-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120029227-A1 METHOD FOR PRODUCING CYCLOPROPANECARBOXYLIC ACID ESTER PCCA, COASY, GRHPR TDP1 4158/4885L3MBTL1 4365/4885LMNA 1488/4885
US-20100305353-A1 METHOD FOR PRODUCING PURIFIED FORMYLCYCLOPROPANE COMPOUND AND INTERMEDIATE OF SUCH FORMYLCYCLOPROPANE COMPOUND FPR1, FPR2, DHPS TDP1 3608/4885L3MBTL1 4207/4885LMNA 4220/4885
US-20100280267-A1 METHOD FOR PRODUCING CYCLOPROPANE CARBOXYLIC ACID COMPOUND AND INTERMEDIATE THEREFOR FAR1, CYP51A1, CYP4A11 TDP1 3924/4885L3MBTL1 3363/4885LMNA 2745/4885
US-20020010361-A1 Process for producing 3,3-dimethyl-2- formylcyclopropane-carboxylic acid ester ACSL6, ACSL3, TRMT1L TDP1 3586/4885L3MBTL1 2566/4885LMNA 4764/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.