SCHEMBL4732880

SCHEMBL4732880

CC(C)c1cc2c(cc1S(=O)(=O)Cl)S(=O)(=O)c1ccccc1C(=O)N2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.37
MEN1 O00255 4/20 0.37
ALDH1A1 P00352 4/20 0.37
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
IGF1R P08069 1/20 0.35
PDGFRB P09619 1/20 0.35
NOX4 Q9NPH5 1/20 0.35
NPC1 O15118 1/20 0.35
MAOA P21397 2/20 0.34
CHEK1 O14757 2/20 0.34
MAPT P10636 1/20 0.34
GPR3 P46089 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HPGD P15428 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CA12 O43570 1/20 0.33
USP2 O75604 1/20 0.33
CA1 P00915 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4732884 0.87 EGFR (0.39) KMT2AMEN1ALDH1A1EGFRERBB2
SCHEMBL4736394 0.85 TGM2 (0.34) CA12CA1CA2CA4CA7
SCHEMBL4737700 0.80 ALDH1A1 (0.40) KMT2AMEN1ALDH1A1MAPTL3MBTL1
SCHEMBL4731530 0.78 BRD4 (0.37) KMT2AMEN1ALDH1A1NPC1MAPT
SCHEMBL4732636 0.76 ACHE (0.44) ALDH1A1MAPTHPGDKDM4E
SCHEMBL4736397 0.76 TGM2 (0.36) EGFRERBB2IGF1RPDGFRBNOX4
SCHEMBL4734512 0.72 BRD4 (0.46) ALDH1A1NPC1MAPTL3MBTL1
SCHEMBL4734516 0.71 DRD2 (0.32) KMT2AMEN1ALDH1A1NPC1MAPT
SCHEMBL4734165 0.70 TAAR1 (0.40) KMT2AMEN1ALDH1A1MAPTL3MBTL1
SCHEMBL5710957 0.69 KMT2A (0.67) KMT2AMEN1ALDH1A1MAOACHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed