SCHEMBL4736394

SCHEMBL4736394

CC(C)c1cc2c(cc1S(=O)(=O)Cl)S(=O)(=O)c1cc(F)ccc1C(=O)N2

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 1/20 0.34
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA4 P22748 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
BACE1 P56817 1/20 0.30
KDR P35968 1/20 0.30
PSEN1 P49768 1/20 0.30
PSEN2 P49810 1/20 0.30
APH1B Q8WW43 1/20 0.30
NCSTN Q92542 1/20 0.30
APH1A Q96BI3 1/20 0.30
PSENEN Q9NZ42 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4736397 0.88 TGM2 (0.36) TGM2BACE1KDRBRD4
SCHEMBL4732880 0.85 KMT2A (0.37) CA12CA1CA2CA4CA7
SCHEMBL4734290 0.80 HTR1A (0.35) BRD4
SCHEMBL4733337 0.79 HTR1A (0.35) BRD4
SCHEMBL4734165 0.79 TAAR1 (0.40)
SCHEMBL4734123 0.77 HTR1A (0.38)
SCHEMBL4735469 0.76 ACHE (0.41) KDR
SCHEMBL4732884 0.76 EGFR (0.39) TGM2
SCHEMBL4737048 0.76 TBXAS1 (0.39)
SCHEMBL4734722 0.75 HCAR3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008061029-A1 ARYL SULFONAMIDE DERIVATIVES AND METHODS OF THEIR USE WYETH (US) 2008-05-22 WO disclosed