SCHEMBL4733778

SCHEMBL4733778

Cc1nc(C(F)F)c(OC(=O)Nc2ccccc2-c2ccc(S(C)(=O)=O)cc2)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
PTGS2 P35354 11/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
DRD1 P21728 1/20 0.36
IKBKB O14920 1/20 0.36
JAK2 O60674 1/20 0.36
JAK3 P52333 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
KDM4E B2RXH2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4733467 0.91 CA2 (0.44) PTGS2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL1019446 0.87 POLB (0.38) ALDH1A1MEN1KMT2AL3MBTL1PTGDR2
SCHEMBL1018834 0.85 CHRM3 (0.44) ALDH1A1GAAJAK2JAK3NPC1
SCHEMBL4731393 0.84 CA2 (0.39) PTGS2NPC1RAB9AMEN1KMT2A
SCHEMBL4733183 0.83 SMN1; SMN2 (0.36) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL1024112 0.81 CHRM3 (0.40) NPC1RAB9AKDM4EMEN1KMT2A
SCHEMBL4733534 0.80 AKR1C3 (0.35) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL4732011 0.80 ALDH1A1 (0.37) ALDH1A1NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL4729048 0.78 RXFP1 (0.35) ALDH1A1MEN1KMT2ARXFP1L3MBTL1
SCHEMBL6255403 0.78 MAPT (0.33) ALDH1A1RAB9AKDM4ESMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008053044-A2 HETARYL CARBON ACID-N-(BIPHEN-2-YL)AMIDE COMPOUNDS BASF SE (DE) 2008-05-08 WO disclosed