SCHEMBL4735834

SCHEMBL4735834

O=C(c1ccnnc1)N(Cc1ccc(Br)nc1)c1ccc(F)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 8/20 0.46
CXCR2 P25025 2/20 0.40
GAA P10253 1/20 0.39
TSHR P16473 1/20 0.39
PDK1 Q15118 2/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
BCL2A1 Q16548 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4737132 0.84 MAPK14 (0.44) MAPK14CXCR2GAATSHRPDK1
SCHEMBL4737075 0.81 MAPK14 (0.40) MAPK14CXCR2PDK1HSP90AA1HSP90AB1
SCHEMBL4735426 0.80 OPRM1 (0.43) MAPK14CXCR2TSHRPDK1
SCHEMBL4737014 0.79 HDAC2 (0.42) MAPK14CXCR2TSHR
SCHEMBL4738924 0.79 OPRM1 (0.40) MAPK14CXCR2TSHR
SCHEMBL4738700 0.78 MAPK14 (0.39) MAPK14CXCR2TSHRPDK1HSP90AA1
SCHEMBL4737305 0.78 DRD4 (0.45) MAPK14CXCR2GAATSHRLMNA
SCHEMBL4733795 0.78 KDM4E (0.51) MAPK14CXCR2TSHRHSP90AB1
SCHEMBL4738909 0.77 TSHR (0.44) MAPK14CXCR2GAATSHRLMNA
SCHEMBL4735517 0.77 MAPK14 (0.38) MAPK14CXCR2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO disclosed