SCHEMBL4736786

SCHEMBL4736786

CCN(CC)c1cccc(CN(C(=O)c2cc3ccccc3s2)c2ccc(Cl)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.41
CNR1 P21554 2/20 0.39
NPY2R P49146 3/20 0.39
CNR2 P34972 2/20 0.38
PDK1 Q15118 1/20 0.38
CYP3A4 P08684 1/20 0.36
HDAC3 O15379 3/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC2 Q92769 3/20 0.36
RAB9A P51151 1/20 0.36
BCL2L1 Q07817 1/20 0.36
GPBAR1 Q8TDU6 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
PIN1 Q13526 1/20 0.35
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8184199 0.81 MAPK14 (0.44) CNR1CNR2PDK1CYP3A4HDAC1
SCHEMBL8190064 0.79 CYP3A4 (0.42) CNR1CNR2PDK1CYP3A4GPBAR1
SCHEMBL4738668 0.77 CNR2 (0.40) CNR1CNR2PDK1CYP3A4GPBAR1
SCHEMBL4733577 0.77 TLR7 (0.40) CNR1CNR2CYP3A4GPBAR1
SCHEMBL4738921 0.76 TRPM8 (0.43) OPRM1NPY2RPDK1HDAC3HDAC1
SCHEMBL3818747 0.76 CNR2 (0.47) CNR1CNR2CYP3A4RAB9A
SCHEMBL4735258 0.76 ALDH1A1 (0.52) CNR2CYP3A4RAB9A
SCHEMBL4739106 0.75 NPC1 (0.41) CNR1CNR2PDK1CYP3A4RAB9A
SCHEMBL3824123 0.74 CNR1 (0.41) CNR1CNR2CYP3A4GPBAR1
SCHEMBL4733672 0.72 ALDH1A1 (0.44) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed