SCHEMBL4738708

SCHEMBL4738708

Cn1cccc1C(=O)N(Cc1ccc(N2CCN(c3ccccn3)CC2)nc1)c1ccc(F)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
CYP1A2 P05177 4/20 0.46
HSD17B10 Q99714 4/20 0.46
CYP2C9 P11712 3/20 0.46
USP2 O75604 2/20 0.46
DRD2 P14416 6/20 0.44
DRD3 P35462 6/20 0.44
DRD4 P21917 4/20 0.44
HTR1A P08908 3/20 0.44
HTR2A P28223 3/20 0.44
HTR7 P34969 3/20 0.44
ADRA2C P18825 1/20 0.44
DRD1 P21728 1/20 0.44
DRD5 P21918 1/20 0.44
HRH1 P35367 1/20 0.44
CYP3A4 P08684 4/20 0.43
SIGMAR1 Q99720 4/20 0.43
CYP2C19 P33261 3/20 0.43
HTR2C P28335 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4803555 0.91 ME2 (0.39) ALDH1A1SMN1; SMN2DRD2DRD3DRD4
SCHEMBL4734210 0.88 HTR1A (0.47) ALDH1A1DRD2DRD3DRD4HTR1A
SCHEMBL4734880 0.87 MEN1 (0.37) ALDH1A1SMN1; SMN2CYP1A2USP2DRD2
SCHEMBL4737954 0.84 KDM4E (0.45) ALDH1A1SMN1; SMN2CYP1A2CYP2C9DRD2
SCHEMBL3065998 0.82 KDM4E (0.46) ALDH1A1SMN1; SMN2CYP1A2HSD17B10CYP2C9
SCHEMBL3826319 0.82 DRD4 (0.47) ALDH1A1SMN1; SMN2CYP1A2CYP2C9DRD2
SCHEMBL4738710 0.82 LMNA (0.49) ALDH1A1SMN1; SMN2CYP1A2HSD17B10CYP2C9
SCHEMBL4737305 0.82 DRD4 (0.45) ALDH1A1SMN1; SMN2CYP1A2CYP2C9DRD2
SCHEMBL4739086 0.82 TSHR (0.52) ALDH1A1SMN1; SMN2CYP1A2CYP2C9DRD2
SCHEMBL4737347 0.80 DRD4 (0.43) ALDH1A1SMN1; SMN2CYP1A2CYP2C9DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed