SCHEMBL4734880

SCHEMBL4734880

Cn1cccc1C(=O)N(Cc1ccc(N2CCN(C(c3ccc(F)cc3)c3ccc(F)cc3)CC2)nc1)c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
ALDH1A1 P00352 2/20 0.37
ME2 P23368 1/20 0.36
ME1 P48163 1/20 0.36
ME3 Q16798 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 1/20 0.36
ACHE P22303 1/20 0.36
CACNA2D1 P54289 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNB1 Q02641 1/20 0.35
CACNA1C Q13936 1/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
DRD1 P21728 1/20 0.35
DRD4 P21917 1/20 0.35
DRD5 P21918 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4803555 0.89 ME2 (0.39) ALDH1A1ME2ME1ME3KDM4E
SCHEMBL4738708 0.87 ALDH1A1 (0.46) ALDH1A1KDM4ETSHRACHEHTR1A
SCHEMBL4734210 0.84 HTR1A (0.47) ALDH1A1ME2ME1ME3KDM4E
SCHEMBL4735318 0.80 OPRM1 (0.37) MEN1KMT2AATMALDH1A1ME2
SCHEMBL4740309 0.80 LMNA (0.46) MEN1KMT2AATMALDH1A1KDM4E
SCHEMBL4736577 0.79 TSHR (0.49) MEN1KMT2AATMALDH1A1KDM4E
SCHEMBL4735549 0.79 MEN1 (0.43) MEN1KMT2AATMALDH1A1KDM4E
SCHEMBL4739217 0.78 MEN1 (0.42) MEN1KMT2AATMALDH1A1ME2
SCHEMBL4735156 0.76 KCNH2 (0.39) ALDH1A1KDM4ETSHRMAPTCYP3A4
SCHEMBL3830332 0.76 MEN1 (0.45) MEN1KMT2AALDH1A1ME2ME1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073461-A2 ION CHANNEL MODULATORS WYETH (US) 2008-06-19 WO claimed