SCHEMBL4744648

SCHEMBL4744648

Cc1cc(O)c2cc(C#N)ccc2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.41
TERT O14746 1/20 0.40
PKM P14618 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
CASP3 P42574 1/20 0.39
KDM1A O60341 1/20 0.39
CSNK1A1 P48729 1/20 0.38
CSNK1D P48730 1/20 0.38
GSK3B P49841 1/20 0.38
CSNK1G2 P78368 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
AR P10275 1/20 0.38
DYRK1A Q13627 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4785913 0.80 LMNA (0.62) PIN1TERTPKMMAPK1SMN1; SMN2
SCHEMBL25830618 0.78 DOT1L (0.49) TERTAR
SCHEMBL5561501 0.78 PIN1 (0.49) PIN1ARDYRK1A
SCHEMBL6205008 0.77 CTSK (0.45) PIN1SMN1; SMN2KDM4EHPGDDYRK1A
SCHEMBL3760247 0.77 LMNA (0.61) SMN1; SMN2KDM4EALDH1A1GAALMNA
SCHEMBL29632523 0.76 NT5E (0.41) PIN1KDM4EARLMNA
SCHEMBL5566519 0.75 CYP11B2 (0.43) PIN1DYRK1A
SCHEMBL3642253 0.74 LMNA (0.41) MAPK1KDM4EALDH1A1GLAGAA
SCHEMBL4966064 0.74 ALDH1A1 (0.55) SMN1; SMN2RXFP1CASP3KDM4EALDH1A1
SCHEMBL4748554 0.74 POLB (0.53) SMN1; SMN2KDM4EALDH1A1LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117079-A1 ANTIMICROBIAL COMPOUNDS BASED UPON 4-AMINOQUINOLINE HELPERBY THERAPEUTICS LIMITED (GB) 2008-10-02 WO disclosed
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed