SCHEMBL476366

SCHEMBL476366

N#Cc1cccc(S(=O)(=O)c2cc(CCNC(=O)O)nn2-c2cccnc2F)c1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 5/20 0.38
GLO1 Q04760 1/20 0.36
SLC40A1 Q9NP59 1/20 0.36
RORC P51449 1/20 0.35
KAT6A Q92794 1/20 0.34
APLNR P35414 1/20 0.34
ROCK2 O75116 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4120239 0.89 HTR6 (0.40) NAMPTALDH1A1L3MBTL1
SCHEMBL4126131 0.88 HTT (0.37) NAMPTALDH1A1L3MBTL1
SCHEMBL476471 0.88 NAMPT (0.35) NAMPTALDH1A1L3MBTL1
SCHEMBL18258908 0.87 NAMPT (0.35) NAMPTKAT6AALDH1A1L3MBTL1
SCHEMBL4137822 0.85 HTR2A (0.39) NAMPTRORCKAT6A
SCHEMBL4139027 0.85 CNR1 (0.39) NAMPTRORC
SCHEMBL476390 0.85 HTT (0.39) NAMPTALDH1A1
SCHEMBL4125767 0.85 NFE2L2 (0.39) NAMPTGLO1SLC40A1
SCHEMBL476373 0.84 GLO1 (0.39) NAMPTGLO1SLC40A1APLNR
SCHEMBL476365 0.84 APLNR (0.35) NAMPTGLO1SLC40A1APLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2412713-B1 PYRAZOLE COMPOUND TAKEDA PHARMACEUTICAL (JP) 2016-11-30 EP disclosed
EP-2412713-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2012-02-01 EP disclosed