SCHEMBL4771067

SCHEMBL4771067

COc1ccc(S(=O)(=O)C2CCN(C(=O)O)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.52
PKM P14618 4/20 0.50
MMP1 P03956 2/20 0.50
MMP8 P22894 2/20 0.50
ALDH1A1 P00352 3/20 0.49
ELOVL6 Q9H5J4 1/20 0.48
TSHR P16473 1/20 0.48
GAA P10253 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MMP2 P08253 2/20 0.47
MMP9 P14780 2/20 0.47
HPGD P15428 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
LMNA P02545 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2928335 0.84 ELOVL6 (0.45) ALDH1A1ELOVL6GAAMEN1KMT2A
SCHEMBL17966724 0.84 MMP13 (0.56) MMP13PKMMMP1MMP8ALDH1A1
SCHEMBL28514815 0.83 STS (0.68) MMP13MMP1MMP8ALDH1A1MMP2
SCHEMBL1807395 0.82 MMP2 (0.49) MEN1KMT2AMMP2MMP9
SCHEMBL28172585 0.82 HTR2A (0.50) MMP13PKMMMP1MMP8ALDH1A1
SCHEMBL4771117 0.82 SPR (0.48) LMNA
SCHEMBL27917812 0.82 HTR2A (0.58) ALDH1A1ELOVL6MEN1KMT2ANPC1
SCHEMBL1188309 0.81 MMP13 (0.73) MMP13PKMMMP1MMP8ALDH1A1
SCHEMBL1809236 0.81 MGLL (0.67) ALDH1A1GAAMEN1KMT2AHPGD
SCHEMBL2634144 0.81 SPR (0.44) TSHRMMP2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107226807-A Tankyrase inhibitor 山东轩竹医药科技有限公司 2017-10-03 CN disclosed
US-7348324-B2 Cyclic amine compounds as CCR5 antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-03-25 US disclosed
EP-1886994-A1 Cyclic amine compounds as CCR5 antagonists Takeda Pharmaceutical Company Limited (JP) 2008-02-13 EP disclosed
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists TOBIRA THERAPEUTICS, INC. 2003-06-19 US disclosed
US-6562978-B1 N-(3-(4-(4-(Aminocarbonyl)benzyl)-1-piperidinyl)propyl)-N-(3, 4-dichlorophenyl)-1-(methylsulfonyl)-4-piperidinecarboxamide or a salt thereof for treatment of AIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-13 US disclosed
EP-1220842-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-10 EP disclosed
WO-2001025200-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists CCR5, CCR1, CCR3 MMP13 4131/4885PKM 4190/4885MMP1 4029/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.