SCHEMBL4774098

SCHEMBL4774098

CN1CCN(C(=O)Cn2c(-c3ccccc3)c(CN3CCC(c4c(F)cccc4F)CC3)c3ccccc32)CC1.Cc1c(CN2CCC(c3c(F)cccc3F)CC2)c2ccccc2n1CC(=O)N1CCN(C)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 2/20 0.41
PTGS2 P35354 1/20 0.40
HTR6 P50406 1/20 0.39
MAPT P10636 2/20 0.39
LMNA P02545 1/20 0.38
GLA P06280 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
EGFR P00533 1/20 0.37
TYMS P04818 1/20 0.37
LTA4H P09960 1/20 0.37
VDR P11473 1/20 0.37
SRC P12931 1/20 0.37
MAPK1 P28482 1/20 0.37
CTSK P43235 1/20 0.37
FABP4 P15090 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4709394 0.96 PTGS2 (0.43) PTGDR2PTGS2HTR6MAPTLMNA
SCHEMBL4708685 0.93 HTR6 (0.43) PTGDR2HTR6MAPTLMNAGLA
SCHEMBL4709041 0.90 PTGS2 (0.40) PTGS2MAPTLMNAEGFRTYMS
SCHEMBL4773925 0.88 POLB (0.42) PTGDR2HTR6MAPTLMNAGLA
SCHEMBL4708187 0.86 CYP3A4 (0.44) PTGS2MAPTEGFRTYMSLTA4H
Trifluoroacetic Acid SCHEMBL4518616 0.85 MAPT (0.42) PTGS2MAPTLMNAGLAL3MBTL1
SCHEMBL4779231 0.84 CNR2 (0.46) PTGDR2LMNAGLAL3MBTL1
SCHEMBL4706301 0.81 KDM4E (0.44) PTGS2MAPTEGFRTYMSLTA4H
SCHEMBL4780894 0.80 LMNA (0.47) PTGDR2MAPTLMNAGLAL3MBTL1
SCHEMBL4776252 0.80 PTGDR2 (0.44) PTGDR2HTR6MAPTTSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008000818-A1 FLUORINATED INDOLEAMIDES USEFUL AS LIGANDS OF THE ORL-1 RECEPTOR BRANE DISCOVERY S.R.L. (IT) 2008-01-03 WO claimed