SCHEMBL4774580

SCHEMBL4774580

O=[N+]([O-])c1ccc(Oc2cc(CCCc3ccccc3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.40
LMNA P02545 3/20 0.39
HTT P42858 2/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
CYP19A1 P11511 2/20 0.38
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
EPHX1 P07099 1/20 0.38
MAPT P10636 2/20 0.37
HPGD P15428 1/20 0.37
MCL1 Q07820 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774683 0.85 NOS3 (0.39) LMNARAB9AMEN1KMT2ASIGMAR1
SCHEMBL4776439 0.79 SPHK1 (0.35) LMNAHTTEPHX1MAPTALDH1A1
SCHEMBL4794914 0.76 ADRA2A (0.45)
SCHEMBL4774754 0.72 PDE5A (0.41) GRIN2BHTTKMT2APOLBCYP19A1
SCHEMBL4780410 0.72 NOS3 (0.44) GRIN2BKMT2APOLBCYP19A1EPHX1
SCHEMBL4779107 0.69 PDE5A (0.47) LMNAHTTKMT2ACYP19A1EPHX1
SCHEMBL4774562 0.69 CYP19A1 (0.42) GRIN2BLMNAMEN1KMT2ASIGMAR1
SCHEMBL4780673 0.68 CYP11B1 (0.45) HTTMEN1KMT2APOLBCYP19A1
SCHEMBL4774100 0.68 NOS3 (0.42) LMNAMEN1KMT2APOLBSIGMAR1
SCHEMBL4778107 0.68 LTB4R (0.48) MEN1KMT2APOLBCYP19A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed