SCHEMBL4776548

SCHEMBL4776548

CC(NC(=N)N)(C(N)=O)c1cccc(-c2nc(CCCc3ccccc3)cc(OCCc3ccccc3)n2)c1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 1/20 0.36
CYP1A2 P05177 1/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CTSS P25774 1/20 0.36
CYP2C19 P33261 1/20 0.36
CTSK P43235 1/20 0.36
KCNH2 Q12809 1/20 0.36
PPARG P37231 5/20 0.35
ALOX5 P09917 5/20 0.35
LTB4R Q15722 6/20 0.35
PTGES O14684 4/20 0.35
PSEN1 P49768 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA1 P30542 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776567 0.78 ALOX5 (0.39) PPARGALOX5LTB4RPTGESPSEN1
SCHEMBL4776562 0.76 MMP2 (0.42) HDAC1HDAC6
SCHEMBL4776784 0.76 C5AR1 (0.37) PPARGALOX5ADORA3ADORA1
SCHEMBL4781761 0.72 LTA4H (0.40) HDAC1HDAC6
SCHEMBL4778137 0.71 ALDH1A1 (0.48) CYP1A2LTB4R
SCHEMBL4778107 0.67 LTB4R (0.48) CYP1A2CYP3A4CYP2C9ALOX5LTB4R
SCHEMBL4780655 0.63 ALDH1A1 (0.46) CYP1A2ALOX5PTGES
SCHEMBL14303803 0.63 MAPT (0.46) CYP2C19
SCHEMBL4796563 0.63 MMP2 (0.46) CYP2C19HDAC1HDAC6
SCHEMBL4778494 0.62 MMP2 (0.45) HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed