SCHEMBL4783994

SCHEMBL4783994

CNS(=O)(=O)c1cc(Nc2cnc(C)c(-n3cc(C(=O)NCC(C)(C)C)nn3)c2)cc(C(C)(C)C)c1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.33
TNNI3K Q59H18 1/20 0.33
DDT P30046 2/20 0.31
MIF P14174 1/20 0.30
ACKR3 P25106 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784000 0.90 DDT (0.34) DDTMIF
SCHEMBL4778554 0.85 DDT (0.42) DDT
SCHEMBL4779207 0.83 NR1I2 (0.38) DDTMIFACKR3
SCHEMBL4782091 0.80 BRAF (0.32) DDT
SCHEMBL4779088 0.79 DDR2 (0.38)
SCHEMBL4780120 0.79 DDR1 (0.35)
SCHEMBL4778561 0.77 DDT (0.45) DDT
SCHEMBL4779210 0.76 TEK (0.41) DDTMIF
SCHEMBL4783774 0.76 NR1I2 (0.36)
SCHEMBL4779766 0.76 NR1I2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed