SCHEMBL479674

SCHEMBL479674

CCOC(=O)COc1cc(Oc2ccc(C(C)C(O)(c3c[nH]c(=O)c(C)c3)C(F)(F)F)c(Cl)c2)ccc1F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPOX P50336 1/20 0.33
DUT P33316 1/20 0.33
THRA P10827 2/20 0.33
THRB P10828 2/20 0.33
ALDH1A1 P00352 4/20 0.32
ESR1 P03372 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
BTK Q06187 1/20 0.31
MAPT P10636 2/20 0.31
HPGD P15428 2/20 0.31
NPSR1 Q6W5P4 2/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
NTSR1 P30989 1/20 0.31
CYP2C19 P33261 1/20 0.31
P2RX3 P56373 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL479790 0.92 MCL1 (0.36) THRATHRBCYP2C19
SCHEMBL479912 0.91 THRB (0.35) THRATHRBBTKMAPTNPSR1
SCHEMBL754455 0.84 PPOX (0.37) PPOXDUTALDH1A1ESR1TDP1
SCHEMBL733146 0.84 PPOX (0.37) PPOXDUTALDH1A1ESR1TDP1
SCHEMBL480263 0.83 PPOX (0.33) PPOXDUTALDH1A1TDP1L3MBTL1
SCHEMBL479958 0.83 MCL1 (0.41) THRATHRBL3MBTL1MAPTSMN1; SMN2
SCHEMBL480020 0.81 PRKAB2 (0.33) P2RX3
SCHEMBL480101 0.81 MCL1 (0.35) THRATHRBALDH1A1
SCHEMBL479931 0.80 S1PR2 (0.33) PPOXTHRATHRBTDP1BTK
SCHEMBL479852 0.80 SMN1; SMN2 (0.40) THRATHRBLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP claimed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO claimed
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed