SCHEMBL4852108

SCHEMBL4852108

CC1(C)CCC(C)(C)N1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FFAR3 O14843 1/20 0.41
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
CYP2C19 P33261 1/20 0.37
APLNR P35414 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16415664 0.97 FFAR3 (0.39) FFAR3TSHRNFKB1CYP2C19
SCHEMBL9067554 0.89 TSHR (0.48) FFAR3TSHRNFKB1CYP2C19
Hydrochloric Acid SCHEMBL11196712 0.87 TSHR (0.47) FFAR3TSHRNFKB1CYP2C19
Ethylene SCHEMBL11463450 0.85 TSHR (0.45) FFAR3TSHRNFKB1CYP2C19
Propene SCHEMBL11410149 0.79 TSHR (0.41) FFAR3TSHRNFKB1CYP2C19
SCHEMBL14369404 0.77 ESR1 (0.41) FFAR3TSHRNFKB1CYP2C19
SCHEMBL22341334 0.74 GAA (0.39)
Lithium Ion SCHEMBL16415663 0.72 FFAR3 (0.32) FFAR3TSHRNFKB1CYP2C19
SCHEMBL30145016 0.70 TSHR (0.38) FFAR3TSHRNFKB1CYP2C19
SCHEMBL6045009 0.70 CYP3A4 (0.42) TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9663546-B2 Metal amides of cyclic amines PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2017-05-30 US disclosed
US-20160152649-A1 METAL AMIDES OF CYCLIC AMINES PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2016-06-02 US disclosed
WO-2015013630-A1 METAL AMIDES OF CYCLIC AMINES PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-01-29 WO disclosed
US-20080149097-A1 Beta-agonist compounds comprising nitric oxide donor groups and reactive oxygen species scavenger groups and their use in the treatment of respiratory disordersB YISSUM RESEARCH DEVELOPMENT COMPANY OF HEBREW UNIVERSITY OF JERUSALEM (IL) 2008-06-26 US disclosed
US-7378438-B2 Beta-agonist compounds comprising nitric oxide donor groups and reactive oxygen species scavenger groups and their use in the treatment of respiratory disorders YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2008-05-27 US disclosed
EP-1503754-B1 BETA-AGONIST COMPOUNDS COMPRISING NITRIC OXIDE DONOR GROUPS AND REACTIVE OXYGEN SPECIES SCAVENGER GROUPS AND THEIR USE IN THE TREATMENT OF RESPIRATORY DISORDERS YISSUM RES DEV CO (IL) 2005-11-23 EP disclosed
US-20050228184-A1 Beta-agonist compounds comprising nitric oxide donor groups and reactive oxygen species scavenger groups and their use in the treatment of respiratory disorders YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2005-10-13 US disclosed
EP-1503754-A1 BETA-AGONIST COMPOUNDS COMPRISING NITRIC OXIDE DONOR GROUPS AND REACTIVE OXYGEN SPECIES SCAVENGER GROUPS AND THEIR USE IN THE TREATMENT OF RESPIRATORY DISORDERS Yissum Research Development Company, of The Hebrew University of Jerusalem (IL) 2005-02-09 EP disclosed
WO-2003088961-A1 BETA-AGONIST COMPOUNDS COMPRISING NITRIC OXIDE DONOR GROUPS AND REACTIVE OXYGEN SPECIES SCAVENGER GROUPS AND THEIR USE IN THE TREATMENT OF RESPIRATORY DISORDERS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 2003-10-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160152649-A1 METAL AMIDES OF CYCLIC AMINES SRM, SMS, NBAS FFAR3 4462/4885TSHR 2429/4885NFKB1 4031/4885
US-20080149097-A1 Beta-agonist compounds comprising nitric oxide donor groups and reactive oxygen species scavenger groups and their use in the treatment of respiratory disordersB ADRA2B, ADRA1B, ADRB1 FFAR3 238/4885TSHR 1485/4885NFKB1 1021/4885
US-20050228184-A1 Beta-agonist compounds comprising nitric oxide donor groups and reactive oxygen species scavenger groups and their use in the treatment of respiratory disorders ADRB1, ADRB2, ADRB3 FFAR3 137/4885TSHR 1366/4885NFKB1 1538/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.