SCHEMBL5206944

SCHEMBL5206944

C#CCn1cc(C2CCN(C(=O)C=Cc3ccccc3)C2)c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.55
MAPT P10636 5/20 0.55
NPC1 O15118 4/20 0.55
SMN1; SMN2 Q16637 4/20 0.55
HPGD P15428 1/20 0.55
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.44
GAA P10253 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CCR2 P41597 2/20 0.42
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4858050 0.82 RAB9A (0.62) RAB9AMAPTNPC1SMN1; SMN2HPGD
SCHEMBL4857604 0.78 MAPT (0.53) RAB9AMAPTNPC1SMN1; SMN2HPGD
SCHEMBL5202233 0.78 HRH2 (0.41) RAB9AMAPTNPC1HPGDALDH1A1
SCHEMBL5205671 0.74 MAPT (0.47) RAB9AMAPTNPC1SMN1; SMN2HPGD
SCHEMBL5203557 0.73 ALDH1A1 (0.50) RAB9AALDH1A1LMNAGAAMEN1
SCHEMBL4849757 0.73 HRH2 (0.47) RAB9AMAPTNPC1SMN1; SMN2ALDH1A1
SCHEMBL4860169 0.70 MAPT (0.40) RAB9AMAPTNPC1SMN1; SMN2HPGD
SCHEMBL7301194 0.69 RAB9A (0.68) RAB9AMAPTNPC1SMN1; SMN2HPGD
SCHEMBL7301191 0.69 RAB9A (0.68) RAB9AMAPTNPC1SMN1; SMN2HPGD
SCHEMBL4858356 0.68 CREBBP (0.42) ALDH1A1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed