SCHEMBL48684

SCHEMBL48684

O=C(O)COCCc1cccc2ccccc12

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.57
KDM4E B2RXH2 3/20 0.53
ALDH1A1 P00352 2/20 0.53
HPGD P15428 1/20 0.53
FFAR4 Q5NUL3 1/20 0.50
CYP1A2 P05177 1/20 0.50
MTNR1A P48039 2/20 0.49
FFAR1 O14842 1/20 0.48
AKR1B1 P15121 1/20 0.48
CDYL Q9Y232 1/20 0.46
MCL1 Q07820 3/20 0.46
CTNNB1 P35222 1/20 0.45
CASP1 P29466 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1180264 0.86 TDP1 (0.56) TDP1KDM4EALDH1A1HPGDFFAR4
SCHEMBL4510057 0.84 TDP1 (0.54) TDP1KDM4EALDH1A1FFAR4CYP1A2
SCHEMBL4795474 0.83 TDP1 (0.61) TDP1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL586305 0.82 CYP1A2 (0.52) TDP1CYP1A2MTNR1AAKR1B1CDYL
Hydrochloric Acid SCHEMBL7275360 0.82 TDP1 (0.59) TDP1KDM4EALDH1A1HPGDCYP1A2
Naphthalene SCHEMBL1848110 0.80 FFAR4 (0.50) TDP1KDM4EALDH1A1HPGDFFAR4
SCHEMBL4564283 0.78 MTNR1A (0.54) TDP1KDM4EALDH1A1HPGDFFAR4
SCHEMBL4521520 0.78 MTNR1A (0.45) TDP1KDM4EALDH1A1FFAR4CYP1A2
SCHEMBL7791197 0.78 FFAR4 (0.48) TDP1KDM4EALDH1A1FFAR4CYP1A2
SCHEMBL1218835 0.78 TDP1 (0.67) TDP1KDM4EFFAR4CYP1A2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE43676-E1 Alkyl ether derivatives or salts thereof TOYAMA CHEMICAL CO., LTD. (JP) 2012-09-18 US disclosed
US-RE43676-E1 Alkyl ether derivatives or salts thereof TOYAMA CHEMICAL CO., LTD. (JP) 2012-09-18 US disclosed
US-8129535-B2 Alkyl ether derivatives or salts thereof TOYAMA CHEMICAL CO., LTD. (JP) 2012-03-06 US disclosed
US-8129535-B2 Alkyl ether derivatives or salts thereof TOYAMA CHEMICAL CO., LTD. (JP) 2012-03-06 US disclosed
US-20090221653-A1 7-(2-amino-1-hydroxy-ethyl)-4-hydroxybenzothiazol-2(3H)-one-derivatives as beta2 adrenoreceptor agonists ASTRAZENECA AB (SE) 2009-09-03 US disclosed
US-20090111992-A1 ALKYL ETHER DERIVATIVES OR SALTS THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-04-30 US disclosed
US-20090111992-A1 ALKYL ETHER DERIVATIVES OR SALTS THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-04-30 US disclosed
US-7468443-B2 Alkyl ether derivatives or salts thereof TOYAMA CHEMICAL CO., LTD. (JP) 2008-12-23 US disclosed
US-7468443-B2 Alkyl ether derivatives or salts thereof TOYAMA CHEMICAL CO., LTD. (JP) 2008-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090221653-A1 7-(2-amino-1-hydroxy-ethyl)-4-hydroxybenzothiazol-2(3H)-one-derivatives as beta2 adrenoreceptor agonists ADRB2, ADRB1, ADRA2C TDP1 4235/4885KDM4E 2699/4885ALDH1A1 243/4885
US-20090111992-A1 ALKYL ETHER DERIVATIVES OR SALTS THEREOF AHNAK, NGF, PMP22 TDP1 3177/4885KDM4E 766/4885ALDH1A1 2334/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.