Cadaverine Tartrate

Cadaverine Tartrate

SCHEMBL4889376

CCOC(=O)[C@@H]1CCCNC1.O=C(O)C(O)C(O)C(=O)O

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3CHRM1CHRM2CHRM3CHRM4ESR1ESR2GABRA1GABRB1GABRG2GBA1HRH1HTR1DHTR2AOPRD1OPRK1OPRM1SLC6A2SLC6A3TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8rplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Cadaverine Tartrate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
SLC6A11 P48066 1/20 0.47
TSHR P16473 1/20 0.47
LMNA P02545 1/20 0.47
SLC6A13 Q9NSD5 1/20 0.47
KDM4E B2RXH2 3/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
ATM Q13315 1/20 0.42
CYP2D6 P10635 1/20 0.42
ALDH1A1 P00352 4/20 0.40
PKM P14618 1/20 0.40
CPN1 P15169 2/20 0.39
CPB2 Q96IY4 2/20 0.39
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cadaverine Tartrate SCHEMBL8198834 1.00 SLC6A1 (0.47) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
Cadaverine Tartrate SCHEMBL6970212 1.00 SLC6A1 (0.47) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
Tartaric Acid SCHEMBL29880655 1.00 SLC6A1 (0.47) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
SCHEMBL132089 0.89 SLC6A1 (0.53) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
SCHEMBL132090 0.89 SLC6A1 (0.53) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
SCHEMBL134525 0.89 SLC6A1 (0.53) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
Hydrochloric Acid SCHEMBL205293 0.88 SLC6A1 (0.52) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
Hydrochloric Acid SCHEMBL5215224 0.88 SLC6A1 (0.52) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
Hydrochloric Acid SCHEMBL22444028 0.88 SLC6A1 (0.52) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA
SCHEMBL14525966 0.85 ALDH1A1 (0.50) SLC6A1SMN1; SMN2SLC6A11TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080182874-A1 Novel Compounds ASTRAZENECA AB (SE) 2008-07-31 US disclosed
US-6569849-B1 N-Substituted azaheterocyclic compounds NOVO NORDISK A/S (DK) 2003-05-27 US disclosed
EP-0934313-B1 N-SUBSTITUTED AZAHETEROCYCLIC COMPOUNDS NOVO NORDISK AS (DK) 2003-05-14 EP disclosed
US-20020151539-A1 Novel heterocyclic compounds JORGENSEN TINE KROGH (DK) 2002-10-17 US disclosed
EP-0851865-B1 12H-Dibenzo[d,g][1,3]dioxocine derivatives NOVO NORDISK AS (DK) 2002-07-17 EP disclosed
US-6391890-B1 ANALGESICS, ANTIINFLAMMATORY AGENTS, NON-INSULIN DEPENDENT DIABETES NOVO NORDISK A/S (DK) 2002-05-21 US disclosed
EP-0869954-B1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF NEUROGENIC INFLAMMATION NOVO NORDISK AS (DK) 2001-09-19 EP disclosed
EP-0820450-B1 N-substituted azaheterocyclic carboxylic acids and alkylesters thereof NOVO NORDISK AS (DK) 2001-09-12 EP disclosed
US-6060468-A ANTIINFLAMMATORY AGENTS NOVO NORDISK A/S (DK) 2000-05-09 US disclosed
US-6054458-A Heterocyclic compounds NOVONORDISKALS (DK) 2000-04-25 US disclosed
EP-0738262-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-23 EP disclosed
WO-1996031499-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed
WO-1996031469-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed
WO-1996031497-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed
WO-1996031471-A1 NOVEL METHOD NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed
EP-0705246-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1996-04-10 EP disclosed
EP-0705248-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1996-04-10 EP disclosed
WO-1995018793-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1995-07-13 WO disclosed
WO-1995000486-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1995-01-05 WO disclosed
WO-1995000483-A1 N-SUBSTITUTED AZAHETEROCYCLIC CARBOXYLIC ACIDS AND ESTERS THEREOF NOVO NORDISK A/S (DK) 1995-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080182874-A1 Novel Compounds REN, F12, GPR119 SLC6A1 928/4885SMN1; SMN2 812/4885SLC6A11 767/4885
US-20020151539-A1 Novel heterocyclic compounds IAPP, GPR119, NPY1R SLC6A1 4566/4885SMN1; SMN2 522/4885SLC6A11 4429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.