SCHEMBL134525

SCHEMBL134525

CCOC(=O)[C@H]1CCCNC1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A1 P30531 2/20 0.53
SLC6A11 P48066 1/20 0.53
TSHR P16473 1/20 0.53
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
SLC6A13 Q9NSD5 1/20 0.53
MAPT P10636 4/20 0.52
KMT2A Q03164 2/20 0.52
KDM4E B2RXH2 1/20 0.52
ATM Q13315 1/20 0.52
CYP2D6 P10635 1/20 0.52
ALDH1A1 P00352 3/20 0.47
PKM P14618 1/20 0.43
MEN1 O00255 1/20 0.43
NOS2 P35228 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL132089 1.00 SLC6A1 (0.53) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
SCHEMBL132090 1.00 SLC6A1 (0.53) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
Hydrochloric Acid SCHEMBL5215224 0.98 SLC6A1 (0.52) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
Hydrochloric Acid SCHEMBL22444028 0.98 SLC6A1 (0.52) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
Hydrochloric Acid SCHEMBL205293 0.98 SLC6A1 (0.52) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
SCHEMBL14525966 0.95 ALDH1A1 (0.50) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
SCHEMBL29295425 0.93 ALDH1A1 (0.53) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
Chloroacetic Acid SCHEMBL27501180 0.91 SLC6A1 (0.49) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
Cadaverine Tartrate SCHEMBL4889376 0.89 SLC6A1 (0.47) SLC6A1SLC6A11TSHRLMNASMN1; SMN2
Cadaverine Tartrate SCHEMBL6970212 0.89 SLC6A1 (0.47) SLC6A1SLC6A11TSHRLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 175 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118184650-A 6- (1H-pyrrolo [2,3-b ] pyridin-3-yl) quinazoline-4-amine derivative, and preparation method and application thereof 中国人民解放军北部战区总医院 2024-06-14 CN claimed
CN-116947879-A BBI608 derivative, preparation method thereof and application thereof in preparing medicines for treating STAT3 mediated diseases 沈阳药科大学 2023-10-27 CN claimed
CN-113402447-B sEH inhibitor or pharmaceutically acceptable composition thereof, and preparation method and application thereof 沈阳药科大学 2022-10-18 CN claimed
US-20260124309-A1 STAT6 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS INC (US) 2026-05-07 US disclosed
US-20260125400-A1 TYK2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS INC (US) 2026-05-07 US disclosed
US-12617797-B2 Substituted pyrazolo [1,5-a]pyrimidines having multimodal activity against pain ESTEVE PHARMACEUTICALS, S.A. (ES) 2026-05-05 US disclosed
US-12534452-B2 N-(1H-imidazol-2-yl)benzamide compound and pharmaceutical composition comprising the same as active ingredient KAINOS MEDICINE, INC. (KR) 2026-01-27 US disclosed
EP-4648851-A1 SUBSTITUTED (HETERO)ANILINES AND THEIR USE Astrazeneca AB (SE) 2025-11-19 EP disclosed
US-20250326732-A1 CHROMEN-2-ONE MODULATORS OF POLRMT PRETZEL THERAPEUTICS, INC. (US) 2025-10-23 US disclosed
EP-4620951-A1 MEMANTINE UREA DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF IN PREPARATION OF MEDICAMENT FOR TREATING SOLUBLE EPOXIDE ENZYME-MEDIATED DISEASES Shenyang Pharmaceutical University (CN) 2025-09-24 EP disclosed
WO-2025149498-A1 BENZYLPIPERIDINE DERIVATIVES AS TRP4 ANTAGONISTS FOR THE TREATMENT OF INFLAMMATORY DISEASES ASTRAZENECA AB (SE) 2025-07-17 WO disclosed
US-20070099934-A1 N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprotein b JANSSEN PHARMACEUTICA N.V. (BE) 2007-05-03 US disclosed
EP-1313725-B1 TRICYCLIC ANTITUMOR COMPOUNDS BEING FARNESYL PROTEIN TRANSFERASE INHIBITORS SCHERING CORP (US) 2007-04-11 EP disclosed
EP-1694644-A2 N-ARYL PIPERIDINE SUBSTITUTED BIPHENYLCARBOXAMIDES AS INHIBITORS OF APOLIPOPROTEIN B JANSSEN PHARMACEUTICA N.V. (BE) 2006-08-30 EP disclosed
WO-2005058824-A2 N-ARYL PIPERIDINE SUBSTITUTED BIPHENYLCARBOXAMIDES AS INHIBITORS OF APOLIPOPROTE IN B JANSSEN PHARMACEUTICA N.V. (BE) 2005-06-30 WO disclosed
US-6127366-A ANTICARCINOGENIC OR ANTITUMOR AGENTS MERCK & CO., INC. (US) 2000-10-03 US disclosed
EP-0862435-A4 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 1999-02-03 EP disclosed
US-5817678-A IMIDAZOLE-CONTAINING PIPERIDINE DERIVATIVES, PEPTIDEMIMETIC MERCK & CO., INC. (US) 1998-10-06 US disclosed
EP-0862435-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1998-09-09 EP disclosed
WO-1997018813-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-05-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260125400-A1 TYK2 DEGRADERS AND USES THEREOF TYK2, CSNK2A1, CSNK2A2 SLC6A1 3746/4885SLC6A11 3929/4885TSHR 256/4885
US-20250326732-A1 CHROMEN-2-ONE MODULATORS OF POLRMT POLRMT, TFAM, POLM SLC6A1 4781/4885SLC6A11 4812/4885TSHR 2586/4885
US-12617797-B2 Substituted pyrazolo [1,5-a]pyrimidines having multimodal activity against pain SIGMAR1, OPRD1, OPRL1 SLC6A1 348/4885SLC6A11 336/4885TSHR 818/4885
US-20260124309-A1 STAT6 DEGRADERS AND USES THEREOF STAT6, NCOR2, NCOR1 SLC6A1 3012/4885SLC6A11 3381/4885TSHR 70/4885
US-20070099934-A1 N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprotein b APOB, PNLIP, LIPC SLC6A1 3895/4885SLC6A11 3590/4885TSHR 2816/4885
US-12534452-B2 N-(1H-imidazol-2-yl)benzamide compound and pharmaceutical composition comprising the same as active ingredient IRAK4, IRAK1, IRAK2 SLC6A1 2120/4885SLC6A11 1826/4885TSHR 762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.