SCHEMBL4963186

SCHEMBL4963186

O=C(O)[C@@H]1CCCN1N1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ACE P12821 7/20 0.40
REN P00797 1/20 0.38
LMNA P02545 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27718628 1.00 ACE (0.40) ACERENLMNACYP2C19HSD17B10
SCHEMBL10905425 0.98 ACE (0.41) ACERENLMNACYP2C19HSD17B10
SCHEMBL16761709 0.96 L3MBTL1 (0.37) ACE
SCHEMBL6528047 0.85 ACE (0.33) ACERENLMNACYP2C19HSD17B10
SCHEMBL3360876 0.84 ACE (0.46) ACERENLMNACYP2C19HSD17B10
SCHEMBL7113056 0.84 ACE (0.46) ACERENLMNACYP2C19HSD17B10
SCHEMBL10905654 0.82 TSHR (0.39) ACEREN
SCHEMBL7850459 0.82 ALDH1A1 (0.41) ACERENHSD17B10
SCHEMBL7694332 0.82 AR (0.35) LMNA
SCHEMBL29586626 0.81 GABRP (0.36) ACEREN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874299-A2 VLA-4 ANTAGONISTS Merck & Co., Inc. (US) 2008-01-09 EP disclosed
WO-2006115918-A2 VLA-4 ANTAGONISTS MERCK & CO., INC. (US) 2006-11-02 WO disclosed