SCHEMBL4977669

SCHEMBL4977669

CN(C)C(=O)c1ccc(-c2ccccc2)c(CCN(c2cccnc2)c2cccnc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.54
CYP11B2 P19099 2/20 0.54
KCNA5 P22460 2/20 0.52
KCNH2 Q12809 1/20 0.48
HTT P42858 1/20 0.40
CYP1A2 P05177 6/20 0.40
CYP3A4 P08684 6/20 0.40
HSD17B10 Q99714 5/20 0.40
ALDH1A1 P00352 3/20 0.40
TSHR P16473 2/20 0.40
TRPV1 Q8NER1 1/20 0.40
GLA P06280 1/20 0.40
CYP2C19 P33261 1/20 0.40
LRRK2 Q5S007 1/20 0.40
ALOX15 P16050 2/20 0.40
CLK4 Q9HAZ1 1/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
PTAFR P25105 2/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4982009 0.87 MKNK1 (0.47) CYP11B1CYP11B2KCNA5KCNH2HTT
SCHEMBL4975675 0.86 MKNK1 (0.47) CYP11B1CYP11B2KCNA5TRPV1PTAFR
SCHEMBL4975764 0.81 CYP46A1 (0.53) ALDH1A1PTAFRMEN1KMT2AROCK2
SCHEMBL4977077 0.81 CYP11B1 (0.53) CYP11B1CYP11B2HTTHSD17B10ALDH1A1
SCHEMBL4975773 0.81 KCNA5 (0.39) CYP11B1CYP11B2KCNA5KCNH2CYP1A2
SCHEMBL4980305 0.78 KCNA5 (0.39) CYP11B1CYP11B2KCNA5KCNH2HTT
SCHEMBL4979253 0.78 CYP11B2 (0.46) CYP11B1CYP11B2KCNA5KCNH2
SCHEMBL4981246 0.77 KMT2A (0.48) CYP11B1CYP11B2KCNA5KCNH2HTT
SCHEMBL4977530 0.76 CYP11B1 (0.48) CYP11B1CYP11B2KCNA5KCNH2CYP3A4
SCHEMBL4979558 0.76 CYP11B2 (0.48) CYP11B1CYP11B2KCNA5KCNH2GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP claimed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO claimed