SCHEMBL5012696

SCHEMBL5012696

[O]c1nc2cccc(N3CCN(CCCCCc4ccc(C(F)(F)F)cc4)CC3)c2s1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.46
HTR1A P08908 11/20 0.44
HTR2C P28335 2/20 0.44
DRD2 P14416 8/20 0.44
HTR2A P28223 8/20 0.44
HTR7 P34969 2/20 0.44
HTR6 P50406 2/20 0.44
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
ADRA1D P25100 1/20 0.41
SLC6A4 P31645 1/20 0.40
HRH1 P35367 1/20 0.40
KCNH2 Q12809 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
DRD1 P21728 1/20 0.40
DRD5 P21918 1/20 0.40
DRD3 P35462 1/20 0.40
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5012698 0.89 SIGMAR1 (0.46) SIGMAR1HTR1AHTR2CDRD2HTR2A
SCHEMBL2091038 0.86 MAOB (0.37) KCNH2
SCHEMBL27666017 0.82 SIGMAR1 (0.49) SIGMAR1HTR1AHTR2CDRD2HTR2A
SCHEMBL5013286 0.79 HTR1A (0.51) SIGMAR1HTR1AHTR2CDRD2HTR2A
SCHEMBL5012728 0.78 SIGMAR1 (0.52) SIGMAR1HTR1AHTR2CDRD2HTR2A
SCHEMBL5011693 0.76 ADRA1A (0.45) SIGMAR1HTR1AHTR2CDRD2HTR2A
SCHEMBL27665886 0.76 SIGMAR1 (0.47) SIGMAR1HTR1AHTR2CDRD2HTR2A
SCHEMBL5016189 0.74 HTR1A (0.49) SIGMAR1HTR1AHTR2CDRD2HTR2A
SCHEMBL2091040 0.74 MAOB (0.37) KCNH2
SCHEMBL5013338 0.73 HRH1 (0.48) HTR1AHTR2CDRD2HTR2AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-B1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMA CO LTD (JP) 2008-10-08 EP disclosed