SCHEMBL5013535

SCHEMBL5013535

O=C1OC2(CCCCC2)N(C(=O)c2sccc2Cl)N1Cc1ccc(F)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
SIGMAR1 Q99720 3/20 0.35
TMEM97 Q5BJF2 2/20 0.35
DRD4 P21917 1/20 0.34
HTT P42858 2/20 0.34
PTGER3 P43115 3/20 0.32
HTR1A P08908 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
NAMPT P43490 1/20 0.32
MAPK8 P45983 1/20 0.32
USP2 O75604 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CACNA1G O43497 2/20 0.31
CACNA1H O95180 2/20 0.31
CACNA1I Q9P0X4 2/20 0.31
PREP P48147 1/20 0.31
KDM4E B2RXH2 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5013588 0.79 HSD11B1 (0.42) ALDH1A1SIGMAR1HTTPTGDR2CACNA1G
SCHEMBL5015096 0.79 KMT2A (0.37) ALDH1A1SIGMAR1TMEM97MAPK8SMN1; SMN2
SCHEMBL5012778 0.76 TP53 (0.37) ALDH1A1SIGMAR1HTTSMN1; SMN2CACNA1G
SCHEMBL1086723 0.74 ALDH1A1 (0.46) ALDH1A1HTR1A
SCHEMBL5016389 0.73 ALDH1A1 (0.35) ALDH1A1SIGMAR1TMEM97HTTPTGER3
SCHEMBL5060789 0.73 PTPN1 (0.41) ALDH1A1TMEM97SMN1; SMN2KDM4E
SCHEMBL5016419 0.72 ALDH1A1 (0.41) ALDH1A1SIGMAR1HTTKDM4E
SCHEMBL5011651 0.69 CHRM2 (0.44) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL5066934 0.67 KMT2A (0.35)
SCHEMBL5011764 0.65 HTT (0.44) ALDH1A1HTTCACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed