SCHEMBL5013588

SCHEMBL5013588

O=C1OC2(CCCCC2)N(C(=O)Cc2ccc(Cl)cc2)N1Cc1ccc(F)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.42
IDO1 P14902 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CACNA1H O95180 4/20 0.35
CACNA1G O43497 2/20 0.35
CACNA1I Q9P0X4 2/20 0.35
SIGMAR1 Q99720 1/20 0.34
SSTR5 P35346 1/20 0.34
HPGD P15428 1/20 0.34
THRB P10828 1/20 0.34
LMNA P02545 1/20 0.34
FFAR2 O15552 1/20 0.33
TBXA2R P21731 1/20 0.33
MDM2 Q00987 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5013535 0.79 ALDH1A1 (0.39) ALDH1A1HTTPTGDR2CACNA1HCACNA1G
SCHEMBL5015096 0.77 KMT2A (0.37) ALDH1A1MEN1KMT2ASIGMAR1LMNA
SCHEMBL5016389 0.77 ALDH1A1 (0.35) ALDH1A1HTTPTGDR2CACNA1HCACNA1G
SCHEMBL5060789 0.76 PTPN1 (0.41) ALDH1A1SSTR5
SCHEMBL5012778 0.76 TP53 (0.37) ALDH1A1HTTKMT2ACACNA1HCACNA1G
SCHEMBL5016419 0.75 ALDH1A1 (0.41) ALDH1A1HTTSIGMAR1LMNA
SCHEMBL1086610 0.72 HSD11B1 (0.47) HSD11B1MEN1KMT2ASSTR5
SCHEMBL5013449 0.68 KAT6A (0.39)
SCHEMBL5011651 0.68 CHRM2 (0.44) ALDH1A1MEN1KMT2ALMNA
SCHEMBL30764735 0.68 HSD11B1 (0.51) HSD11B1ALDH1A1HTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed