SCHEMBL5015096

SCHEMBL5015096

O=C1OC2(CCCCC2)N(C(=O)c2cc(C(F)(F)F)ccc2Cl)N1Cc1ccc(F)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.37
MAPK8 P45983 1/20 0.35
MAPK10 P53779 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 1/20 0.35
TSHR P16473 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
P2RX7 Q99572 1/20 0.35
CRHR1 P34998 2/20 0.34
MRGPRX4 Q96LA9 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
TMEM97 Q5BJF2 1/20 0.34
CCR2 P41597 2/20 0.34
LMNA P02545 1/20 0.34
PARP1 P09874 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5060789 0.79 PTPN1 (0.41) ALDH1A1P2RX7TMEM97SMN1; SMN2
SCHEMBL5013535 0.79 ALDH1A1 (0.39) MAPK8ALDH1A1SIGMAR1TMEM97SMN1; SMN2
SCHEMBL5013588 0.77 HSD11B1 (0.42) KMT2AALDH1A1MEN1SIGMAR1LMNA
SCHEMBL1086126 0.76 KMT2A (0.41) KMT2AMAPK8MAPK10MRGPRX4SMN1; SMN2
SCHEMBL5012778 0.74 TP53 (0.37) KMT2AALDH1A1SIGMAR1LMNASMN1; SMN2
SCHEMBL5011835 0.73 CYP1A2 (0.43) ALDH1A1LMNA
SCHEMBL5016389 0.73 ALDH1A1 (0.35) ALDH1A1TSHRL3MBTL1SIGMAR1TMEM97
SCHEMBL5016419 0.70 ALDH1A1 (0.41) ALDH1A1TSHRL3MBTL1P2RX7SIGMAR1
SCHEMBL5011651 0.67 CHRM2 (0.44) KMT2AALDH1A1MEN1TSHRL3MBTL1
SCHEMBL5011764 0.67 HTT (0.44) KMT2AALDH1A1MEN1TSHRL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed