SCHEMBL5016389

SCHEMBL5016389

CC(C)(CC(=O)O)C(=O)N1N(Cc2ccc(F)c(F)c2)C(=O)OC12CCCCC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HTT P42858 2/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTGDR2 Q9Y5Y4 2/20 0.35
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
RIPK1 Q13546 1/20 0.33
KDM4E B2RXH2 1/20 0.32
RAB9A P51151 1/20 0.32
CACNA1H O95180 2/20 0.32
SIGMAR1 Q99720 2/20 0.32
CACNA1G O43497 1/20 0.32
CACNA1I Q9P0X4 1/20 0.32
PTGER3 P43115 3/20 0.31
DRD3 P35462 1/20 0.31
TMEM97 Q5BJF2 1/20 0.31
PTGER4 P35408 1/20 0.31
PTGFR P43088 1/20 0.31
PTGER2 P43116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5016419 0.77 ALDH1A1 (0.41) ALDH1A1HTTTSHRL3MBTL1LMNA
SCHEMBL5013588 0.77 HSD11B1 (0.42) ALDH1A1HTTPTGDR2LMNACACNA1H
SCHEMBL5012778 0.76 TP53 (0.37) ALDH1A1HTTLMNARAB9ACACNA1H
SCHEMBL5013535 0.73 ALDH1A1 (0.39) ALDH1A1HTTPTGDR2KDM4ERAB9A
SCHEMBL5015096 0.73 KMT2A (0.37) ALDH1A1TSHRL3MBTL1LMNASIGMAR1
SCHEMBL5060789 0.69 PTPN1 (0.41) ALDH1A1KDM4ETMEM97
SCHEMBL5066934 0.67 KMT2A (0.35) LMNA
SCHEMBL5011747 0.64 KCNK3 (0.40) ALDH1A1LMNA
SCHEMBL5011764 0.64 HTT (0.44) ALDH1A1HTTTSHRL3MBTL1LMNA
SCHEMBL5011651 0.64 CHRM2 (0.44) ALDH1A1TSHRL3MBTL1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910381-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-04-16 EP disclosed
WO-2007000325-A2 SUBSTITUTED 1-OXA-3,8-DIAZASPIRO[4.5]-DECAN-2-ON- COMPOUNDS AND THE USE THEREOF FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-01-04 WO disclosed