SCHEMBL5015216

SCHEMBL5015216

COc1cc(N(C)C(=O)N(C)c2[c]cccc2)cc(OC)c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 4/20 0.38
LMNA P02545 3/20 0.38
MAPT P10636 3/20 0.38
MAPK1 P28482 2/20 0.38
GFER P55789 1/20 0.38
MCL1 Q07820 1/20 0.38
TUBB1 Q9H4B7 3/20 0.38
TUBB4A P04350 2/20 0.38
TUBB P07437 2/20 0.38
TUBA3C P0DPH7 2/20 0.38
TUBA1B P68363 2/20 0.38
TUBA4A P68366 2/20 0.38
TUBB4B P68371 2/20 0.38
TUBB3 Q13509 2/20 0.38
TUBB2A Q13885 2/20 0.38
TUBB8 Q3ZCM7 2/20 0.38
TUBA3E Q6PEY2 2/20 0.38
TUBA1A Q71U36 2/20 0.38
TUBA1C Q9BQE3 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3790835 0.72 CYP2C9 (0.47) ALDH1A1LMNAMAPTTSHRCYP1A2
SCHEMBL2535686 0.70 TSHR (0.42) ALDH1A1LMNAMAPTMAPK1PKM
SCHEMBL7480109 0.69 MAPT (0.45) KDM4EALDH1A1LMNAMAPTMAPK1
SCHEMBL95841 0.68 ALDH1A1 (0.39) KDM4EALDH1A1MAPTTDP1SMN1; SMN2
SCHEMBL16294301 0.68 RAB9A (0.36) KDM4E
SCHEMBL21305541 0.68 MEN1 (0.43) KDM4EALDH1A1TSHRL3MBTL1
SCHEMBL1416233 0.67 ALOX5 (0.34) ALDH1A1MAPTTDP1SMN1; SMN2TSHR
SCHEMBL482524 0.64 KMT2A (0.45) KDM4EALDH1A1LMNASMN1; SMN2HTT
SCHEMBL27995633 0.64 KDM4E (0.45) KDM4EALDH1A1MAPTMAPK1TUBB1
SCHEMBL1416613 0.64 ROCK2 (0.35) ALDH1A1LMNAPKMSMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1138673-B1 Novel carbamates and ureas as modifiers of multi-drug resistance VERTEX PHARMA (US) 2008-08-06 EP claimed