Asparagine

Asparagine

SCHEMBL50255

NC(=O)C[C@H](N)C(=O)O.O

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Asparagine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 known ✓ P39086 7/20 0.52
GRIK2 known ✓ Q13002 4/20 0.52
PTGS1 known ✓ P23219 1/20 0.48
GRIA4 known ✓ P48058 4/20 0.45
GRIK3 known ✓ Q13003 4/20 0.45
GRIK5 known ✓ Q16478 4/20 0.45
GRIA2 known ✓ P42262 3/20 0.44
GRIA1 known ✓ P42261 2/20 0.44
GRIA3 known ✓ P42263 1/20 0.44
GRIN2A known ✓ Q12879 1/20 0.44
ALOX15 P16050 1/20 0.54
BLM P54132 1/20 0.54
PMP22 Q01453 1/20 0.54
KMT2A Q03164 1/20 0.54
GRM1 Q13255 2/20 0.52
GRM2 Q14416 2/20 0.52
SLC7A5 Q01650 1/20 0.50
SLC7A11 Q9UPY5 1/20 0.48
GGT1 P19440 4/20 0.46
SLC1A1 P43005 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Asparagine SCHEMBL28655930 1.00 ALOX15 (0.54) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL29449905 1.00 ALOX15 (0.54) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL656714 1.00 ALOX15 (0.54) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL28655929 1.00 ALOX15 (0.54) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL8103410 1.00 ALOX15 (0.54) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL656713 1.00 ALOX15 (0.54) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL50254 1.00 ALOX15 (0.54) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL28196111 0.97 ALOX15 (0.52) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL31634581 0.97 ALOX15 (0.52) ALOX15BLMPMP22KMT2AGRIK1
Asparagine SCHEMBL150535 0.97 ALOX15 (0.56) ALOX15BLMPMP22KMT2AGRIK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2012 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122012373-A CHO-K1 cell chemistry limiting basic culture medium 华北制药集团新药研究开发有限责任公司 2026-05-12 CN claimed
EP-4017496-B1 FORMULATIONS FOR USE IN THE PREVENTION AND/OR TREATMENT OF PERIPHERAL NEUROPATHY AND ITS ASSOCIATED DISEASES LOH YIN SZE (SG) 2026-01-07 EP claimed
US-12359164-B2 Process for producing cell culture media MERCK PATENT GMBH (DE) 2025-07-15 US claimed
CN-120005806-A CHO cell culture medium and application thereof 江苏埃美益生物技术有限公司 2025-05-16 CN claimed
CN-119307441-B Culture solution of bovine cloned embryo and application thereof 内蒙古大学 2025-03-21 CN claimed
CN-119307441-A Culture solution of bovine cloned embryo and application thereof 内蒙古大学 2025-01-14 CN claimed
CN-119265134-A System, method and organoid suitable for organ/organoid circulatory culture 苏州先觉生物科技有限公司 2025-01-07 CN claimed
CN-119020257-A Perfusion culture medium for mammalian CHO cells and application thereof 信达生物制药(苏州)有限公司 2024-11-26 CN claimed
EP-4455263-A1 COMPOSITION FOR CULTURING ANIMAL CELLS AJINOMOTO CO., INC. (JP) 2024-10-30 EP claimed
EP-3192368-B1 COMPOSITION FOR PRESERVING CELLS, CONTAINING, AS ACTIVE INGREDIENTS, PLANT-DERIVED RECOMBINANT HUMAN SERUM ALBUMIN AND PLANT PEPTIDES CEFO CO LTD (KR) 2024-10-30 EP claimed
EP-0994657-B1 PALATABLE ELEMENTAL MEDICAL FOOD ABBOTT LAB (US) 2004-01-28 EP claimed
US-6245803-B1 ENTERAL ADMINISTERING NUTRIENTS ABBOTT LABORATORIES 2001-06-12 US claimed
EP-0780469-B1 Immortalized human skin cell lines and serum-free medium for the production thereof NESTLE SA (CH) 2001-02-28 EP claimed
EP-1059352-A1 Long term cell culture of human carcinoma Oncodia AG (CH) 2000-12-13 EP claimed
EP-0994657-A1 PALATABLE ELEMENTAL MEDICAL FOOD Abbott Laboratories (US) 2000-04-26 EP claimed
US-5922766-A NUTRITIONALLY COMPLETE FOR HUMANS WITH SPECIALIZED DIETARY NEEDS, USES SPECIFIC FREE AMINO ACIDS TO PROVIDE THE SOUCE OF AMINO NITROGEN(PROTEIN EQUIVALENTS) AND SPECIAL BLENDS OF FATS THAT PROVIDE PLEASANT TASTING FORMULA WITH CALORIES ABBOTT LABORATORIES 1999-07-13 US claimed
WO-1999001044-A1 PALATABLE ELEMENTAL MEDICAL FOOD ABBOTT LABORATORIES (US) 1999-01-14 WO claimed
WO-1995012664-A1 ADAPTION OF MAMMALIAN CELL LINES TO HIGH CELL DENSITIES GENETICS INSTITUTE, INC. (US) 1995-05-11 WO claimed
US-5326908-A Process for the preparation of asparagine NSC TECHNOLOGIES LLC 1994-07-05 US claimed
EP-0162422-A2 The novel physiologically active substance foroxymithine, a process and microorganisms for its production and its use as medicament MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1985-11-27 EP claimed