SCHEMBL5070401

SCHEMBL5070401

COc1c(N)c(-c2ccccc2)cc(C)c1C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.37
FEN1 P39748 2/20 0.37
PDE4B Q07343 4/20 0.37
PDE4A P27815 3/20 0.37
PDE4C Q08493 3/20 0.37
PDE4D Q08499 3/20 0.37
IKBKB O14920 1/20 0.36
HSD17B10 Q99714 2/20 0.35
FYN P06241 1/20 0.35
SQOR Q9Y6N5 1/20 0.35
KCNA3 P22001 1/20 0.34
ACHE P22303 1/20 0.34
BACE1 P56817 1/20 0.33
TSHR P16473 1/20 0.33
ESR2 Q92731 1/20 0.33
MAPT P10636 2/20 0.32
PTGS2 P35354 1/20 0.32
MET P08581 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2680108 0.81 PDE4B (0.42) ALOX5APFEN1PDE4BPDE4APDE4C
SCHEMBL27833081 0.73 PDE4B (0.44) ALOX5APFEN1PDE4BPDE4APDE4C
SCHEMBL14674863 0.70 MET (0.45) BACE1MET
SCHEMBL22025913 0.69 PDE4B (0.47) PDE4BPDE4APDE4CPDE4DHSD17B10
SCHEMBL2203934 0.68 FYN (0.50) PDE4BPDE4APDE4CPDE4DFYN
SCHEMBL2202989 0.68 ACHE (0.40) IKBKBHSD17B10ACHEBACE1TSHR
SCHEMBL2849367 0.68 ACHE (0.40) IKBKBHSD17B10ACHEBACE1TSHR
SCHEMBL9326316 0.68 ALDH1A1 (0.54) PDE4BPDE4APDE4CPDE4DIKBKB
SCHEMBL12325398 0.67 PDE4B (0.56) PDE4BPDE4APDE4CPDE4DIKBKB
SCHEMBL1903608 0.67 PDE4B (0.49) PDE4BPDE4APDE4CPDE4DIKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942904-A2 CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITORS Merck & Co., Inc. (US) 2008-07-16 EP disclosed
WO-2007041494-A2 CHOLESTERYL ESTER TRANSFER PROTEIN INHIBITORS MERCK & CO., INC. (US) 2007-04-12 WO disclosed