SCHEMBL5082809

SCHEMBL5082809

CS(=O)(=O)O.C[C@H](NCCc1ccccc1)C(=O)c1ccccc1

nearest known ligand 0.48

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.48
MEN1 O00255 2/20 0.48
OPRK1 P41145 1/20 0.48
TSHR P16473 1/20 0.48
ALDH1A1 P00352 4/20 0.47
SIGMAR1 Q99720 3/20 0.47
GAA P10253 2/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
CYP3A4 P08684 1/20 0.47
BLM P54132 1/20 0.47
GFER P55789 1/20 0.47
PMP22 Q01453 1/20 0.47
AKR1C3 P42330 1/20 0.47
HPGD P15428 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5082438 0.94 SIGMAR1 (0.53) KMT2AMEN1OPRK1TSHRALDH1A1
SCHEMBL5082242 0.88 NPC1 (0.46) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL5079098 0.87 NPC1 (0.43) KMT2AMEN1OPRK1TSHRALDH1A1
SCHEMBL5082682 0.86 MAOB (0.51) SIGMAR1MAPTLMNAHPGDHDAC2
SCHEMBL5082447 0.86 MAOB (0.51) SIGMAR1MAPTLMNAHPGDHDAC2
SCHEMBL5079910 0.86 NPC1 (0.43) KMT2AMEN1OPRK1TSHRALDH1A1
SCHEMBL5076506 0.85 OPRK1 (0.62) KMT2AMEN1OPRK1TSHRSIGMAR1
SCHEMBL8093031 0.85 KMT2A (0.56) KMT2AALDH1A1SIGMAR1HPGDCYP2D6
Hydrochloric Acid SCHEMBL5082431 0.85 NPC1 (0.43) KMT2AMEN1OPRK1TSHRALDH1A1
Hydrochloric Acid SCHEMBL8092291 0.84 KMT2A (0.55) KMT2AMEN1ALDH1A1SIGMAR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7408084-B2 Process for producing optically active β-amino alcohol KANEKA CORPORATION (JP) 2008-08-05 US disclosed
US-20050277791-A1 Process for producing optically active beta-amino alcohol KANEKA CORPORATION (JP) 2005-12-15 US disclosed
EP-1512677-A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE s-AMINO ALCOHOL KANEKA CORPORATION (JP) 2005-03-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050277791-A1 Process for producing optically active beta-amino alcohol ADH1A, ALDH7A1, ADH1C KMT2A 1460/4885MEN1 3339/4885OPRK1 21/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.