SCHEMBL5096401

SCHEMBL5096401

N#CCc1nc(NCCc2ccc(O)cc2)ncc1-c1nc2ccccc2s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ILK Q13418 4/20 0.48
CDK1 P06493 1/20 0.45
KDR P35968 1/20 0.45
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
MAPT P10636 3/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
MAPK9 P45984 2/20 0.41
MAPK10 P53779 2/20 0.41
MAPK8 P45983 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
IRAK4 Q9NWZ3 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5103181 0.91 ALDH1A1 (0.43) ILKCDK1KDRNPC1RAB9A
SCHEMBL5596244 0.91 CDK1 (0.43) ILKCDK1KDRNPC1RAB9A
SCHEMBL5103578 0.88 SMN1; SMN2 (0.46) CDK1KDRNPC1RAB9AMAPT
SCHEMBL5110395 0.86 ALDH1A1 (0.46) ILKCDK1KDRNPC1RAB9A
SCHEMBL17709604 0.86 MAPK10 (0.56) ILKCDK1KDRNPC1RAB9A
SCHEMBL5138885 0.84 CSNK1D (0.41) ILKCDK1KDRNPC1RAB9A
SCHEMBL5100115 0.84 PTGS1 (0.41) ILKCDK1KDRNPC1RAB9A
SCHEMBL5596497 0.84 KDM4E (0.42) ILKCDK1KDRNPC1RAB9A
SCHEMBL5596747 0.79 CDK1 (0.35) ILKCDK1KDRNPC1RAB9A
SCHEMBL5103679 0.76 IRAK4 (0.46) KDRIRAK4MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7470686-B2 Method of inhibiting the expression and/or the activity of JNK LABORATOIRES SERONO SA (CH) 2008-12-30 US claimed