SCHEMBL510481

SCHEMBL510481

O=Cc1ccc(SCc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.53
MAOB P27338 3/20 0.53
SLC6A4 P31645 1/20 0.49
ALDH1A1 P00352 2/20 0.48
CYP2A6 P11509 1/20 0.48
PPARG P37231 2/20 0.45
PPARA Q07869 2/20 0.45
HAO1 Q9UJM8 1/20 0.45
ALOX5 P09917 1/20 0.45
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
DAO P14920 1/20 0.41
POLB P06746 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LTA4H P09960 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL510243 0.92 MEN1 (0.49) MAOAMAOBSLC6A4ALDH1A1CYP2A6
SCHEMBL5043419 0.83 CA12 (0.56) MAOAMAOBALDH1A1CYP2A6ALOX5
SCHEMBL2294886 0.81 ALDH5A1 (0.57) MAOAMAOBALDH1A1KDM4EMEN1
SCHEMBL20704671 0.81 CYP2A6 (0.57) ALDH1A1CYP2A6KDM4EMEN1KMT2A
SCHEMBL21331846 0.81 ALDH1A1 (0.61) MAOAMAOBALDH1A1MEN1KMT2A
SCHEMBL13695939 0.81 ALDH5A1 (0.57) MAOAMAOBALDH1A1KDM4EMEN1
SCHEMBL19631194 0.81 MAOA (0.53) MAOAMAOBSLC6A4ALDH1A1PPARG
SCHEMBL10480960 0.81 PIM1 (0.58) MAOAMAOBMEN1KMT2APOLB
SCHEMBL10480959 0.81 PIM1 (0.58) MAOAMAOBMEN1KMT2APOLB
SCHEMBL1710689 0.80 MAOA (0.49) MAOAMAOBSLC6A4ALDH1A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 116 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210093691-A1 Glycopeptide Compounds Having Activity Of Resisting Drug-Resistant Bacteria, And Preparation Method And Application Thereof SHANGHAI LAIYI CENTER FOR BIOPHARMACEUTICAL R&D CO., LTD. (CN) 2021-04-01 US claimed
EP-3763728-A1 GLYCOPEPTIDE COMPOUNDS HAVING ACTIVITY OF RESISTING DRUG-RESISTANT BACTERIA, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shanghai LaiYi Center For Biopharmaceutical R&D Co., Ltd. (CN) 2021-01-13 EP claimed
CN-107129451-B Novel belt cyano diphenylethyllene sulfosalt preparation method and applications 同济大学 2019-12-03 CN claimed
WO-2019170046-A1 GLYCOPEPTIDE COMPOUNDS HAVING ACTIVITY OF RESISTING DRUG-RESISTANT BACTERIA, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 上海来益生物药物研究开发中心有限责任公司 2019-09-12 WO claimed
CN-107129451-A Novel belt cyano group diphenylethyllene sulfosalt preparation method and applications 同济大学 2017-09-05 CN claimed
US-5808164-A Process for producing aromatic sulfides PHILLIPE PETROLEUM COMPANY (US) 1998-09-15 US claimed
US-20250367173-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME LIGACHEM BIOSCIENCES INC (KR) 2025-12-04 US disclosed
EP-4540245-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME LigaChem Biosciences Inc. (KR) 2025-04-23 EP disclosed
CN-119654323-A External nucleotide pyrophosphatase-phosphodiesterase-1 inhibitor and pharmaceutical composition containing the same 瑞嘉化学生物科学股份有限公司 2025-03-18 CN disclosed
CN-119192236-B Serine hydrolase inhibitor and preparation method and application thereof 西北农林科技大学深圳研究院 2025-03-11 CN disclosed
CN-119192236-A Serine hydrolase inhibitor and preparation method and application thereof 西北农林科技大学深圳研究院 2024-12-27 CN disclosed
WO-2023242631-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME LEGOCHEM BIOSCIENCES, INC. (KR) 2023-12-21 WO disclosed
WO-2023242631-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME LEGOCHEM BIOSCIENCES, INC. (KR) 2023-12-21 WO disclosed
US-5120754-A Anticholesterol and antidiabetic agents PFIZER INC. (US) 1992-06-09 US disclosed
US-5061717-A ANTICHOLESTEROL AGENTS PFIZER INC. (US) 1991-10-29 US disclosed
EP-0383281-A1 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same TOYAMA CHEMICAL CO., LTD. (JP) 1990-08-22 EP disclosed
WO-1989008650-A1 THIAZOLIDINEDIONE HYPOGLYCEMIC AGENTS PFIZER INC. (US) 1989-09-21 WO disclosed
EP-0332331-A2 Thiazolidinedione hypoglycemic agents PFIZER INC. (US) 1989-09-13 EP disclosed
EP-0089154-A2 Ethanolamine derivatives, their preparation and use in pharmaceutical compositions BEECHAM GROUP PLC (GB) 1983-09-21 EP disclosed
US-4399075-A Process for producing chlorinated phenoxytoluene derivatives ASAHI CHEMICAL COMPANY, LIMITED (JP) 1983-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250367173-A1 ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME ENPP1, ENPP3, SMPD1 MAOA 724/4885MAOB 828/4885SLC6A4 2583/4885
US-20210093691-A1 Glycopeptide Compounds Having Activity Of Resisting Drug-Resistant Bacteria, And Preparation Method And Application Thereof VIP, CUTA, MGAM MAOA 2941/4885MAOB 2702/4885SLC6A4 4536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.